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3-{1-[(4-methylpiperazin-1-yl)sulfonyl]piperidin-3-yl}benzoic acid
5-benzyl-4-(4-methyl-1H-imidazole-2-carbonyl)-1-(4-methylphenyl)piperazin-2-one
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amine
4-{1-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-1H-imidazol-2-yl}quinoline
(1S,4S)-2-(2-{3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}ethyl)-2-azabicyclo[2.2.1]heptane
3-{5-[2-(benzyloxy)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
1-methyl-3-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}-1H-indole
1-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]-4-(2-phenylethyl)piperazine
N-[3-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)carbamoyl}amino)phenyl]-N-methylacetamide
1-(1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-yl)-2-methylpiperidine
2-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-[2-(4-methanesulfonylphenyl)pyrimidin-4-yl]pyrrolidin-3-ol
5-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-N-(2-methoxyethyl)-1-methyl-1H-1,3-benzodiazol-2-amine
3-[5-(1-benzylpiperidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridazine
(1r,4r)-4-{[benzyl(2-hydroxyethyl)amino]methyl}cyclohexan-1-ol
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-3-(1H-pyrazol-1-yl)benzamide
8-chloro-N-[(2R)-pyrrolidin-2-ylmethyl]quinoline-2-carboxamide
5-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-[4-(2-chlorophenoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-(4-methoxyphenyl)-2,2-dimethyl-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperazine
1-(2,6-dimethoxypyridine-3-carbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
(3S,4S)-1-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-4-methylpiperidine-3,4-diol
3-(4-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)phenol
2-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-4-yl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-cyclopropyl-3-{1-[1-(4-fluorophenyl)propan-2-yl]piperidin-4-yl}propanamide
5-oxo-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)pyrrolidine-3-carboxylic acid
N-[(5-ethylpyridin-2-yl)methyl]-6-methyl-2-(morpholin-4-yl)pyrimidin-4-amine
5-(3,4-dimethoxybenzoyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(1S,5R)-6-(4-fluoro-3-methoxybenzoyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-3-cyclobutanecarbonyl-6-(4,6-dimethylpyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-methoxy-2-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-1,4-dihydropyridin-4-one
3-(2-ethyl-1H-imidazol-1-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
5-(1H-1,3-benzodiazole-5-carbonyl)-N-cyclopentyl-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-tert-butyl-4-hydroxy-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]pyrimidine-5-carboxamide
8-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3S,4R)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
(1-methyl-5-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
(3S,4R)-1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-4-phenylpyrrolidine-3-carboxylic acid
5-({3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}methyl)-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-[1-(carbamoylmethyl)-1H-imidazol-2-yl]-N-[2-(thiophen-2-yl)ethyl]piperidine-1-carboxamide
1-tert-butyl-4-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}pyrrolidin-2-one
2,6-dimethyl-4-{[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}phenyl acetate
4-hydroxy-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-2-(pyridin-2-yl)pyrimidine-5-carboxamide
2-{[1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
6-(4-ethylphenyl)-N-[2-(1H-pyrazol-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-[(5-chloro-2,4-dimethoxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[3-(2-ethoxyethoxy)benzoyl]-2-(4-fluorophenyl)morpholine
3-fluoro-4-methoxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
N-(butan-2-yl)-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-(pyridin-4-ylmethyl)acetamide