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3-(1H-imidazol-1-ylmethyl)-1-(5-methyl-4-phenylthiophene-3-carbonyl)piperidine
N-(1,4-oxazepan-6-ylmethyl)azepane-1-sulfonamide
N-[3-(4-methylpiperazin-1-yl)butyl]-2-(phenylamino)pyrimidine-5-carboxamide
1-benzyl-3-methyl-8-[(1-methyl-1H-indol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,4S)-4-[(9H-fluoren-2-ylmethyl)(methyl)amino]oxolan-3-ol
4-[(2-chlorophenyl)methyl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
({5-[(4-chlorophenyl)sulfanyl]furan-2-yl}methyl)(methyl)[1-(pyrimidin-4-yl)ethyl]amine
(2R,6S)-1-(oxan-4-ylmethyl)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[1-(pyrazin-2-yl)piperidin-3-yl]-3-(pyridin-3-yl)propanamide
5-(1-{[5-(4-methoxyphenyl)furan-2-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
[3-(2-methoxyethyl)-1-(1,2,3,4-tetrahydroquinoline-8-carbonyl)piperidin-3-yl]methanol
1-(1-{6-[(furan-3-ylmethyl)amino]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
3-chloro-4-[(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)oxy]-N-(2-methoxyethyl)benzamide
2-(3,5-dichloropyridin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
1-(2-{[(3,4-dimethylphenyl)carbamoyl]amino}ethyl)piperidine-3-carboxamide
1-(4-{[3-(2,3-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenyl)-1H-1,2,4-triazole
7-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2,5-dimethylpyrazolo[1,5-a]pyrimidine
3-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)propanamide
N-methyl-4-({2-methyl-2,7-diazaspiro[4.5]decan-7-yl}methyl)benzene-1-sulfonamide
6-(2-aminoethyl)-2-methyl-N-[2-(pyrrolidin-1-yl)ethyl]pyrimidin-4-amine
N-[2-(1H-imidazol-1-yl)ethyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
N-{[3-(dimethylamino)thiolan-3-yl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
6-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)imidazo[1,2-a]pyridine-2-carboxamide
1,3-dimethyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-[(4-amino-6-{[(5-methylpyrazin-2-yl)methyl]amino}pyrimidin-2-yl)sulfanyl]-N,N-dimethylacetamide
4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}thiomorpholine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-(2-oxopyrrolidin-1-yl)butanamide
1-ethoxy-3-{[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}propan-2-ol
2-amino-4-[3-(2-hydroxyethoxy)phenyl]-6-(2-methoxyphenyl)pyridine-3-carbonitrile
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propan-2-yl)piperidine
3-({8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)benzonitrile
6-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-N-(propan-2-yl)pyrimidin-4-amine
(2S)-1-[(2-chloro-5-ethoxy-4-propoxyphenyl)methyl]pyrrolidine-2-carboxamide
3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1-[3-(2-methylpyrimidin-4-yl)phenyl]urea
7,8-dimethyl-4-(piperidine-1-carbonyl)-2-(1-propyl-1H-pyrazol-4-yl)quinoline
(2S,4S)-4-amino-N-(propan-2-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]pyrrolidine-2-carboxamide
4-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-4-(4-methylphenoxy)piperidine
3-(1-methyl-1H-pyrrol-2-yl)-N-(piperidin-4-yl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
4-chloro-1-[2-(4-cyclopropanecarbonyl-3-fluorophenyl)ethyl]-1H-pyrazole
1-[(4-fluorophenyl)methyl]-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
7-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-2-oxa-7-azaspiro[4.5]decane
3-{[(diphenylmethyl)amino]methyl}-7-fluoro-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-N'-(2,4,6-trimethylphenyl)butanediamide
ethyl 4-{3-[2-(cyclohexylformamido)ethyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}piperidine-1-carboxylate
N-[(5-methylthiophen-2-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
(1R,5R)-N,N-dimethyl-6-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
6-acetyl-2-amino-4-[1-(pyridin-4-yl)-1H-pyrrol-2-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile