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1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-2-phenylazetidine
4-(1,3-benzothiazol-2-yl)-2-(thiomorpholin-4-ylmethyl)phenol
N-methyl-4-oxo-4-phenyl-N-[(1-phenylpyrrolidin-3-yl)methyl]butanamide
2-[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-(furan-2-ylmethyl)acetamide
2-{4-[4-(3-methoxypiperidin-1-yl)piperidin-1-yl]phenyl}-1-(pyrrolidin-1-yl)ethan-1-one
2-methyl-N-{[1-(prop-2-en-1-yl)pyrrolidin-3-yl]methyl}-6-(propan-2-yl)pyrimidin-4-amine
N-(2-oxoazepan-3-yl)-5-phenoxyfuran-2-carboxamide
(2-{2-[1-(3,4-dimethylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
2-(dimethyl-1,3-thiazol-5-yl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
3-{5-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-(oxolan-2-ylmethoxy)ethan-1-one
(1S,5R)-3-[(1-ethyl-1H-indol-5-yl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
1-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]-3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propan-1-one
(4aS,8aR)-1-(2-phenylethyl)-6-(pyridazine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(4-methoxyphenoxy)piperidine
9-(4-fluorobenzoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
5-[2-(6-methylpyridin-2-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(2S,4S)-4-amino-1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidine-2-carboxylic acid
{7-chloro-5-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
5-(5-chloronaphthalen-1-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-{[4-(cyclohexylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-4-methoxyphenol
N,6,6-trimethyl-5-oxo-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}thiomorpholine-3-carboxamide
(1S,5R)-3-[(4-chlorophenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{[1-(thiophen-3-ylmethyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
4-({2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)benzonitrile
1-(2,3-dihydro-1H-inden-2-yl)-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,4-diazepane
4-(2,4-dimethoxyphenyl)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole
2-(4,5-dimethyl-1H-imidazol-1-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
1-(2-methoxyphenyl)-5-(oxan-2-yl)-3-(propan-2-yl)-1H-1,2,4-triazole
3-{4-[6-amino-5-cyano-4-(1-methyl-1H-pyrazol-4-yl)pyridin-2-yl]-3,5-dimethyl-1H-pyrazol-1-yl}propanoic acid
3-(2,4-dichloro-3-methylphenyl)-1-[3-(4-methylpiperazin-1-yl)butyl]urea
N-[2-(ethanesulfonyl)ethyl]-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)(thiophen-3-ylmethyl)amine
3-(benzenesulfonyl)-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl)[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
4-(1H-imidazol-2-yl)-1-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidine
2-[(3-methoxyphenyl)methyl]-8-(3,3,4,4-tetrafluorobutyl)-2,8-diazaspiro[4.5]decan-3-one
3-(3-fluorophenyl)-5-(furan-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-(1,4-dioxan-2-ylmethyl)-N-methyl-3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-(thiophen-3-yl)pyridin-2-amine
2-{[4-(3-chloropyridin-2-yl)piperazin-1-yl]methyl}benzonitrile
(2S)-2-(hydroxymethyl)-N-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-pyrazol-5-yl)pyrrolidine-1-carboxamide
5-({methyl[(3-phenyl-1H-pyrazol-4-yl)methyl]amino}methyl)pyrimidin-2-amine
6-methyl-5-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-2-oxo-1,2-dihydropyridine-3-carbonitrile
1-(4-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
{1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-4-yl}(thiophen-2-yl)methanol
propan-2-yl 4-chloro-3-({[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]carbamoyl}amino)benzoate
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
2-{4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}pyridine-3-carbonitrile
3-(2-methoxyethyl)-5-[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]-1-propyl-1H-1,2,4-triazole