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4-[6-amino-5-cyano-4-(3-ethyl-1,2-oxazol-5-yl)pyridin-2-yl]benzoic acid
1-(carbamoylmethyl)-N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]piperidine-3-carboxamide
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(4-fluorophenyl)-1,4-diazepane
1-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-4-(pyrimidin-2-yl)-1,4-diazepane
2-{3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-1,3-thiazole-4-carboxamide
2-(3,3-difluoropiperidin-1-yl)-4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidine
N-(butan-2-yl)-9-oxo-N-(thiophen-3-ylmethyl)-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
4-(dimethyl-1,3-oxazole-5-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1S,5R)-6-(pyridin-2-ylmethyl)-3-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(3-{[(4-fluorophenyl)methyl]sulfanyl}propyl)-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)benzamide
N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-N-(3-phenylprop-2-yn-1-yl)cyclopropanamine
N-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-N-(pyridin-4-ylmethyl)cyclopropanamine
1-(2-methoxyphenyl)-4-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)piperazin-2-one
3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-6-methoxy-1,2-dihydroquinolin-2-one
2-{1-[1-(thian-4-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-amine
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}but-3-en-1-one
4-(methoxymethyl)-6-(3,4,5-trimethoxyphenyl)pyrimidine
6-[(diethylamino)methyl]-N-[(3S)-2-oxoazepan-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-{2-[1-(7-methyl-1-benzofuran-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
7-methoxy-3-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
5-(1H-indol-1-ylmethyl)-N-[1-(3-methylpyridin-2-yl)propyl]-1H-pyrazole-3-carboxamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
1-({4-[1-(cyclohexylmethyl)-1H-1,2,4-triazol-5-yl]phenyl}methyl)-4-methylpiperazine
(2S)-2-amino-1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pentan-1-one
N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-methyl-N-(pyridin-4-ylmethyl)piperidin-4-amine
3,5-dimethyl-1-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}-1H-pyrazole
3-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindole-2-carbonyl]-1,2-dihydroquinoxalin-2-one
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]propan-1-one
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-{[1-(1H-imidazole-5-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
3-[(3R,4S)-4-(dimethylamino)-1-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]piperidin-3-yl]propanoic acid
1-[2-(4-methoxyphenyl)ethyl]-5-(4-methyl-1H-imidazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-(4-methoxyphenyl)-N-{[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]methyl}acetamide
2-ethyl-6-{1-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
(1S,6R)-9-(2-methyl-1,8-naphthyridine-3-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
(2S,4R)-4-amino-N-ethyl-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}pyrrolidine-2-carboxamide
1-(5-methyl-1,3-oxazole-4-carbonyl)-3-(4-methylphenoxymethyl)piperidine
1-{1-[4-(2-methyl-1H-imidazol-4-yl)phenyl]ethyl}piperidine
3-chloro-4-{[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]oxy}-N-cyclopentylbenzamide
ethyl 1-(7-chloroquinolin-4-yl)-5-{[(furan-2-ylmethyl)amino]methyl}-1H-pyrazole-4-carboxylate
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-2-(methylsulfanyl)acetamide
7-(cyclopropylmethyl)-2-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(3-chlorophenyl)methyl]-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-amine
4-(1H-pyrazole-3-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 2-(3-oxo-1-{[3-(prop-2-en-1-yl)-4-(propan-2-yloxy)phenyl]methyl}piperazin-2-yl)acetate
1-cyclohexyl-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-benzyl-4-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,4-diazepan-6-ol
5-[3-(5-methylfuran-2-yl)-1-propyl-1H-1,2,4-triazol-5-yl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxylic acid