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3-[({3-[2-hydroxy-3-(piperidin-1-yl)propoxy]-4-methoxyphenyl}methyl)amino]-2,2-dimethylpropan-1-ol
4-(2-amino-6-methylpyrimidin-4-yl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
7-[(2,3-difluorophenyl)methyl]-2-[3-(methylsulfanyl)propyl]-2,7-diazaspiro[4.5]decane
[(2-butoxy-3-methoxyphenyl)methyl][(6-chloropyridin-3-yl)methyl]amine
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(diethylamino)ethan-1-one
5-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-phenyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[2-methoxy-5-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
{[2-(2-methylphenoxy)pyridin-3-yl]methyl}(pyridin-3-ylmethyl)amine
2-methyl-4-phenyl-9-(pyridin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-(2-amino-6-methylpyrimidin-4-yl)-N-(6-cyanopyridin-3-yl)piperazine-1-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}propanamide
3-{[(6-aminopyridin-3-yl)carbamoyl]methyl}-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-(2-methoxyethyl)-1-methyl-N-(pyridin-2-ylmethyl)azepane-2-carboxamide
1-methyl-9-[8-(trifluoromethyl)quinolin-4-yl]-1,4,9-triazaspiro[5.5]undecan-5-one
methyl 4-{4-[3-(thiophen-3-yl)propanoyl]piperazin-1-yl}benzoate
3-methyl-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
7-[(3,5-dichlorophenyl)methanesulfonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[cyclohexyl(methyl)amino]-3-{2-[(2,2-dimethylmorpholin-4-yl)methyl]phenoxy}propan-2-ol
3-methanesulfonyl-N-(2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
1-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-5-oxopyrrolidine-3-carboxylic acid
6-(5-ethylthiophene-3-carbonyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
3-(2-phenylethyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-oxazole-5-carboxamide
(1R,3s,6r,8S)-4-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-azatricyclo[4.3.1.13,8]undecane
3-({2-[1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
methyl 8-[(4-acetamidophenyl)methyl]-1-(2-methoxyethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-(1H-1,3-benzodiazol-1-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
2-{4-[(2-chlorophenyl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-fluoro-6-methoxy-N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}benzamide
7-(1-ethyl-1H-pyrazole-3-carbonyl)-N2,N2,N4,N4-tetramethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-(pyridin-2-ylmethyl)acetamide
N-{2-[(dimethylcarbamoyl)methyl]phenyl}-2-(1,3-thiazol-2-yl)pyrrolidine-1-carboxamide
2-{8-chloro-[1,2,4]triazolo[4,3-a]pyridin-3-yl}pyridine
4-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
3-(4-chlorophenyl)-N-[2-(4,6-dihydroxypyrimidin-2-yl)ethyl]-3-phenylpropanamide
(3R,5S)-N3-(4-fluorophenyl)-N5-(naphthalen-1-ylmethyl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
[(3R,4R)-1-(2-methyl-1,3-thiazole-4-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
5-methyl-2-{[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1H-1,3-benzodiazole
[1-({1-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
(1S,3R)-3-amino-N-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)cyclopentane-1-carboxamide
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-methylphenyl)ethan-1-one
5-({[(5-ethylpyridin-2-yl)methyl](methyl)carbamoyl}amino)-2-methoxy-N,N-dimethylbenzamide
1-(azocan-1-yl)-3-[5-methoxy-2-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-(2,2-dimethyloxan-4-yl)-5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methylimidazo[1,2-a]pyridine-6-carboxamide
4-(1-butyl-1H-imidazol-2-yl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
4-[2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-1λ6-thiomorpholine-1,1-dione
N-(3-fluorophenyl)-2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidine-6-carboxamide
1-[2-(1H-imidazol-1-yl)-1-phenylethyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea