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pyridin-2-yl(1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)methanol
N-methyl-N-(propan-2-yl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
1-[(1R,5R)-6-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(quinoline-2-carbonyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
(1R,2R,6S,7S)-N-[2-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
5-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-1-methyl-1,2-dihydropyridin-2-one
2-[4-(2-aminophenyl)-1H-pyrazol-1-yl]-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]acetamide
1-(2,6-dimethylpyridin-4-yl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperazine
1-[3-(1-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1H-imidazol-2-yl)phenyl]ethan-1-one
2-(ethylamino)-N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}pyrimidine-5-carboxamide
(2S,4S)-4-amino-N-(propan-2-yl)-1-(pyridine-4-carbonyl)pyrrolidine-2-carboxamide
N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-2-(morpholin-4-yl)-2-oxoacetamide
N,N-dimethyl-5-{[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenoxyethan-1-one
(4aS,7aR)-N-(3-cyanophenyl)-6,6-dioxo-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-[3-(4-methylphenyl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-benzoyl-4-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]piperazine
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
(3R,5S)-5-(morpholine-4-carbonyl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-propyl-1H-pyrazole-5-carboxamide
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
4-{[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
(1S,5R)-6-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
7-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-[({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)methyl]-6-methoxy-1,2-dihydroquinolin-2-one
methyl 3-{[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]carbamoyl}propanoate
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methylacetamide
[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)(thiophen-2-ylmethyl)amine
N'-methyl-N'-phenyl-N-{2-[4-(propan-2-yl)morpholin-2-yl]ethyl}ethanediamide
N-[(1-ethyl-1H-indazol-3-yl)methyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
3-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(5-methylpyrazin-2-yl)methyl]benzamide
3-(2-methoxyacetamido)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]benzamide
1-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
8-[(2-ethoxyphenyl)methyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
4-chloro-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-propanamidobenzamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
2-[1-(thiophen-3-ylmethyl)piperidin-2-yl]pyridine
(2S,4R)-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)-1-[(2,3,4-trimethoxyphenyl)methyl]pyrrolidine-2-carboxamide
2-ethyl-4-{[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]methyl}pyrimidine
N-(2-methoxyethyl)-2,5,7-trimethyl-N-(thiophen-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-yl)pyrrolidin-3-ol
N-cyclopentyl-5-(1H-indole-3-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(2-methylphenoxy)-1-(pyridin-2-ylmethyl)piperidine-4-carboxylic acid
N-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
5-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
3,3-dimethyl-1-[(3S,4R)-1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-4-(propan-2-yl)pyrrolidin-3-yl]urea