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2-ethyl-4-methyl-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-1,3-thiazole-5-carboxamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-(2H-1,3-benzodioxol-5-yl)propan-1-one
3-{2-[({4-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)amino]ethyl}-1,3-oxazolidin-2-one
(3S)-N,N-dimethyl-1-[1-(pyridine-3-carbonyl)piperidin-4-yl]azepan-3-amine
methyl 6-methyl-2-(4-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperazin-1-yl)pyrimidine-4-carboxylate
7-(2-hydroxyethyl)-2-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one
5-methyl-1-{[1-(3-methylpyridin-2-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(2-methoxyethyl)-8-(oxan-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-[2-(propan-2-yl)phenyl]-3-{pyrazolo[1,5-a]pyridin-3-ylmethyl}urea
N-(4-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)pyrazolo[1,5-a]pyridine-7-carboxamide
2-{1-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]piperidin-4-yl}ethan-1-ol
3-(2-methoxypyridin-3-yl)benzonitrile
2-({1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
3-[5-(4-chloro-1,3-dimethyl-1H-pyrazol-5-yl)-1,2,4-oxadiazol-3-yl]pyridazine
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-3-yl]methanol
4,4,4-trifluoro-1-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]butan-1-one
1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-(2,3-difluoro-6-methoxybenzoyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
4-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-6-(propan-2-yloxy)pyrimidin-2-amine
N-(1H-1,2,3-benzotriazol-4-yl)-4-(oxan-4-yl)piperazine-1-carboxamide
N-(1-benzylpyrrolidin-3-yl)-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
1-({1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}methyl)-1H-1,2,3,4-tetrazole
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(3-methylthiophen-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(3-methyl-1-benzothiophene-2-carbonyl)-2-(pyrrolidine-1-carbonyl)piperazine
2-(furan-2-yl)-5-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}pyrimidine
1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-(3-methoxyphenyl)piperidine
2-amino-6-(3,4-difluorophenyl)-4-(1,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N'-(2,4-dimethylphenyl)-N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]propanediamide
2-{[3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]amino}-N-(pyrazin-2-yl)acetamide
(2S,4S)-4-amino-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-N,N-diethylpyrrolidine-2-carboxamide
4-methyl-2-{1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
3-(2-methyl-1H-1,3-benzodiazol-1-yl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]propan-1-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-fluorobenzamide
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-3-[(oxan-4-yl)amino]-5-[(propan-2-yl)sulfamoyl]benzamide
7-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-N,N-dimethylazepan-4-amine
2-(dimethylamino)-N-[2-(dimethylamino)-1-phenylethyl]-N,4-dimethylpyrimidine-5-carboxamide
1-{4-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-4-oxobutyl}pyrrolidin-2-one
1-{2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-[(4-fluorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-[(3-chloro-1-benzothiophen-2-yl)methyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(1-methylcyclopropanecarbonyl)piperidin-3-yl]piperazine
N-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2,3-dihydro-1,4-benzodioxine-6-carboxamide
(4aS,8aR)-1-butyl-6-[3-(pyridin-4-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
2-{3-[3-(5-ethylpyrimidin-2-yl)phenyl]-1H-pyrazol-1-yl}-1-(morpholin-4-yl)ethan-1-one
[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl][1-(1H-imidazol-1-yl)propan-2-yl]amine
8-(1,3-benzothiazol-2-yl)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,8-diazaspiro[4.5]decane
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-(isoquinolin-5-ylmethyl)-N-methylpiperidine-3-carboxamide
(3R,4R)-1-(5,6-dimethylpyrazin-2-yl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol