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(3S,4S)-4-(propan-2-yl)-1-(4,4,4-trifluorobutanoyl)pyrrolidine-3-carboxylic acid
3-(azocan-1-yl)-N-[3-(cyclohexyloxy)-2-hydroxypropyl]propanamide
2-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,2-oxazolidine
N-(2,2-dimethyloxan-4-yl)-N-ethyl-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
2-cyano-N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]benzamide
8-(2-ethylpyridine-4-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-ethyl-3-(piperidin-4-ylmethyl)-1-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(1H-imidazol-1-ylmethyl)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidine
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
2-ethyl-4-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-1-(propan-2-yl)piperazine
11-{[(4-fluorophenyl)methyl]amino}-4-(3-methoxypropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
5-ethyl-N-(3-hydroxypropyl)-4-(pyrrolidin-1-ylmethyl)-N-(thiophen-2-ylmethyl)furan-2-carboxamide
1-(cyclohexylmethyl)-5-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]piperidin-4-amine
3-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
N,6-dimethyl-2-(quinolin-3-yl)pyrimidin-4-amine
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
N-[2-(dimethylamino)ethyl]-2-methyl-N-(oxolan-2-ylmethyl)furan-3-carboxamide
1-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-4-cyclopropanecarbonyl-1,4-diazepan-6-ol
(2R)-N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}oxolane-2-carboxamide
1-[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-2-(methoxymethyl)piperidine
N-[(3R,4S)-1-[(3-chloro-4-methoxyphenyl)methyl]-4-cyclopropylpyrrolidin-3-yl]-3-hydroxypropanamide
2-benzyl-N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1,3-thiazole-4-carboxamide
1-[(3-chlorophenyl)methyl]-3-methyl-5-(1H-1,2,3-triazol-1-ylmethyl)-1H-1,2,4-triazole
2-({2-cyclopentyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-N-cyclopropylacetamide
7-cyclohexyl-2-(2,6-dimethylpyrimidine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3S,4R)-1-[2-(naphthalen-2-yloxy)acetyl]-4-propylpyrrolidin-3-yl]acetamide
3-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanoic acid
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-hydroxyethan-1-one
2-(5-fluoro-2-methyl-1H-indol-3-yl)-1-[4-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]ethan-1-one
2-chloro-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]pyridine-4-carboxamide
4-{4-[(5-cyclopentylthiophen-2-yl)methyl]piperazin-1-yl}-6-methylpyrimidin-2-amine
1-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-3-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
3-{1-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-1H-1,2,3-triazol-4-yl}phenol
2-benzyl-8-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
5-fluoro-2-{3-[1-(oxolan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine
4-chloro-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
6-[2-(dimethylamino)phenyl]-N2,N2-dimethylpyrimidine-2,4-diamine
N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-2-(1-methylpiperidin-2-yl)acetamide
2-cyclopropyl-1-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1H-imidazole
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}pyrazine-2-carboxamide
3-ethyl-N-[(4-hydroxyphenyl)methyl]-4-methyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
N-(3-methoxyphenyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carboxamide
4-(1-benzyl-1H-imidazol-2-yl)-1-(butane-1-sulfonyl)piperidine
N-[2-(4-ethylphenoxy)ethyl]-N-methyl-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-[2-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-oxoethyl]-4,6-dimethyl-1,2-dihydropyrimidin-2-one
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-4-(1H-pyrazol-3-yl)benzamide
2-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}pyridine
1-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-(2-methyl-5-sulfamoylphenyl)urea
(2S,4S)-4-amino-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]pyrrolidine-2-carboxylic acid