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3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-(1H-pyrrole-2-carbonyl)piperidine
1-(3-methanesulfonamidophenyl)-3-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
3-({[1-(oxane-4-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
1-[2-(2,4-dichlorophenoxy)acetyl]azetidine-2-carboxylic acid
(3S,5R)-1-(oxan-4-yl)-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
3-[2-(dimethylamino)ethyl]-8-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 3-{[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]methyl}benzoate
6-(2H-1,3-benzodioxol-5-yl)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyridine-3-carboxamide
4-[3-(1H-imidazol-2-yl)benzoyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-methyl-4-{3-methyl-5-[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]-1H-1,2,4-triazol-1-yl}piperidine
(4aR,7aS)-1-ethyl-4-[(4-phenyl-1,3-thiazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-(2-methylpyridin-4-yl)-1,4-diazepane
1'-(1,3-dimethyl-1H-pyrazole-4-carbonyl)spiro[indene-1,4'-piperidine]
3-(3-chlorobenzoyl)-1-[(3,5-dimethoxyphenyl)methyl]piperidine
5-[4-(diphenylmethyl)piperazin-1-yl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
1-(5-methylthiophene-2-carbonyl)-4-(2-phenoxyethyl)-1,4-diazepan-5-one
1-(3-methoxypropyl)-8-[3-(5-methylfuran-2-yl)butyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-chloro-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}pyridine-2-carboxamide
(2S)-4-methyl-2-{[5-(naphthalen-2-yl)-1,2,4-triazin-3-yl]amino}pentanamide
5-{2-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(oxolan-2-ylmethyl)-N-{[4-(thiophen-2-ylmethoxy)phenyl]methyl}cyclohexanecarboxamide
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-2-(1H-1,2,3-triazol-1-yl)acetamide
4-benzyl-3-{1-[3-(1H-imidazol-4-yl)propanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1-methanesulfonylpiperidin-3-yl)piperazine
4-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-[(4-fluorophenyl)methyl]morpholine
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3,4-dimethoxybenzene-1-sulfonamide
N-ethyl-5-[3-(2-methoxyethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]pyrimidin-2-amine
2-(2-methylpropyl)-4-oxo-N-[2-(propan-2-yl)phenyl]-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxamide
1-(1-{1-[(2,6-difluorophenyl)methyl]piperidin-4-yl}ethyl)-4-methylpiperazine
N-[(1S)-2-(1H-imidazol-4-yl)-1-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl]acetamide
8-(cyclopropylmethyl)-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-(1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-1-oxobutan-2-yl)-2,3-dihydro-1H-isoindol-1-one
4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholine
2-{5-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]-1H-pyrazol-3-yl}phenol
2-amino-1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-methylpropan-1-one
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-[2-(methylsulfanyl)ethyl]pyridin-2-amine
2-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
N3-[(5-methylfuran-2-yl)methyl]-N5-[(4-methylphenyl)methyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
5-(4-methyl-1H-imidazol-2-yl)-1-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-4-phenyl-1H-imidazole
(1S,5R)-6-(pyridin-2-ylmethyl)-3-[3-(thiophen-2-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(4-fluorophenyl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
5-{1-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]piperidin-4-yl}-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
1-(4-{6-oxa-9-azaspiro[4.5]decan-9-ylmethyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
N-(1H-indol-2-ylmethyl)-1-(5-propylpyrimidin-4-yl)piperidin-4-amine
1-[4-({[(dimethyl-1,3-thiazol-2-yl)methyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(2-fluorophenyl)methyl]-5-({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)azepan-2-one
4-[(2-{1-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}-1H-imidazol-1-yl)methyl]pyridine
1-[3-(1H-imidazol-2-yl)benzoyl]-4-(4-methoxyphenoxy)piperidine