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1-ethyl-3-(2-methylpropyl)-N-[1-(pyrazin-2-yl)piperidin-4-yl]-1H-pyrazole-5-carboxamide
6-chloro-2-(2-cyclopropylpyrimidin-5-yl)-N-methyl-N-(propan-2-yl)quinoline-4-carboxamide
(1R,7S)-6-(4,4-difluoropiperidine-1-carbonyl)-3-(2-ethoxyethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}cyclobutanecarboxamide
N-{2-[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-methyl-1,3-thiazole-4-carboxamide
(1R,5R)-3-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-[(2S)-1-methoxypropan-2-yl]-3-[(4-methyl-1,4-diazepan-1-yl)sulfonyl]benzamide
1-[2-methoxy-4-(thiomorpholin-4-ylmethyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
8-{[1-(2-methylphenyl)-1H-pyrrol-2-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]propanamide
5-(1-{2H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}pyrrolidin-2-yl)-N-(2-methoxyethyl)thiophene-2-carboxamide
ethyl 4-[7-chloro-3-({N-cyclopropyl-1-[4-(trifluoromethyl)phenyl]formamido}methyl)quinolin-2-yl]piperazine-1-carboxylate
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-ethyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
1-(4-{[(3-cyclopentylpropyl)amino]methyl}-2-methoxyphenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
N-[2-(1H-imidazol-4-yl)ethyl]-3-(1H-pyrazol-4-yl)benzamide
6-(1H-indol-5-yl)-N,N-dimethylpyridine-2-carboxamide
methyl 3-{[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylformamido]methyl}-5-(4-fluorobenzenesulfonamido)benzoate
N-propyl-4-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-sulfonyl)benzamide
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-3-methylbut-2-en-1-one
5-[(adamantan-1-ylmethyl)(methyl)amino]-1-[(2-fluorophenyl)methyl]azepan-2-one
4-[(4-chloro-3-fluorophenyl)methyl]-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]piperazin-2-one
2-(5-ethylthiophene-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-[(1S,5R)-6-[2-(3,5-difluorophenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
2-chloro-5-acetamido-N-[(2-methylphenyl)(pyridin-4-yl)methyl]benzamide
methyl 4-{[(4aR,8aS)-1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-decahydro-1,6-naphthyridin-6-yl]methyl}benzoate
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[(2-methoxy-5-methylphenyl)carbamoyl]methyl}propanamide
4-{2-[(2-chlorophenyl)methyl]morpholine-4-carbonyl}-N-methylpyridin-2-amine
1-ethyl-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(2H-1,3-benzodioxol-5-yl)-1-{3-[benzyl(methyl)amino]piperidin-1-yl}ethan-1-one
8-[2-amino-6-(propan-2-yl)pyrimidine-4-carbonyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2,3-dihydro-1H-inden-2-yl)-3-[2-(methylsulfanyl)ethyl]-5-(1,3-thiazol-4-ylmethyl)-1H-1,2,4-triazole
methyl (2S)-2-{[1-(4,7-dimethylquinazolin-2-yl)piperidin-4-yl]formamido}-2-phenylacetate
2-(1H-1,3-benzodiazol-2-ylmethoxy)-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
N-butyl-2-(2,6-dioxo-1,3-diazinan-1-yl)-N-[(4-methylphenyl)methyl]acetamide
5-[1-(4-fluorophenyl)cyclopropanecarbonyl]-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
2-amino-4-(3-ethenylphenyl)-6-(pyrazine-2-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-(2-methoxyethyl)-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-methyl-3-[3-(2-methylpropyl)-1-phenyl-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
2-({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}(methyl)amino)ethan-1-ol
8-(2-ethoxyethyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
4-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-2-(trifluoromethyl)morpholine
1-[2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-3-phenylpiperidine
2-[(3-methoxyphenyl)methyl]-8-[2-(morpholin-2-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
ethyl 3-[(3-methoxyphenyl)methyl]-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxylate
6-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1H-indole
N-[1-(4-fluorophenyl)ethyl]-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
4-{[6-(2,5-dimethoxyphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-1,4-oxazepane
1-[2-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-oxoethyl]-2-methyl-1,4-dihydroquinolin-4-one