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1-(cyclopropylmethyl)-4-(3-methyl-1H-pyrazole-5-carbonyl)-2-(propan-2-yl)-1,4-diazepane
5-[3-(oxan-4-yl)-1-(quinoxalin-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
2-[5-(methoxymethyl)thiophene-2-carbonyl]-1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
methyl 1-(3-{3-[(cyclobutylamino)methyl]phenoxy}-2-hydroxypropyl)piperidine-4-carboxylate
3-(4-tert-butylbenzoyl)-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
N-[(4-methylphenyl)(pyridin-4-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-benzyl-8-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 2-(1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)acetate
3-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-indazole
5-(azepane-1-carbonyl)-1-(butan-2-yl)-4-oxo-N-[2-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
N-({1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
2-[2-(trifluoromethyl)benzenesulfonyl]-2,7-diazaspiro[4.5]decane
N-(2-phenoxyethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-(4-methylpentyl)-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
methyl[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
N-[2-(3-methoxyphenyl)-1-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]ethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
4-hydroxy-N-[2-(N-methylmethanesulfonamido)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(3S,4S)-1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-4-(naphthalen-2-yl)piperidin-3-ol
1-[4-({[2-(1H-imidazol-4-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
9-(1-benzofuran-5-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
N-[(3-methoxyphenyl)methyl]-1-methyl-N-(prop-2-en-1-yl)azepane-2-carboxamide
2-methyl-4-[(2S)-2-phenylbutyl]-1-(propan-2-yl)piperazine
6-[2-(pyridin-3-yloxy)propyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-[3-(2-fluorophenoxy)azetidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
6-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-N,N-dimethylpyrazine-2-carboxamide
(3S,4S)-1-[4-(3-hydroxy-3-methylbutyl)benzoyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
(3S,4S)-1-(3-methyl-1,2-oxazole-5-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
N-[(2S)-4-methyl-1-oxo-1-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}pentan-2-yl]acetamide
2-cyclopentyl-1-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
4-chloro-1-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-indazole
6-[2-(furan-2-yl)azepane-1-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)pyridine-3-carboxamide
2-{4-[(3,4-dimethylphenyl)methyl]-3-oxopiperazine-1-carbonyl}pyrrolidine-1-carboxamide
1-(3-chloro-4-propoxyphenyl)-3-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]urea
(1S,5R)-N-(2-fluorophenyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N6-(3-methoxypropyl)-N5-methyl-N5-[3-(morpholin-4-yl)propyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-({1-[4-(methylsulfanyl)butan-2-yl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
2-[4-(dimethylamino)phenyl]-1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
6-[3-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
2-[2-(1H-imidazol-4-yl)ethyl]-8-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-sulfamoylbenzamide
1-{2-[(4aR,8aR)-4a-hydroxy-7-(pyrimidin-2-yl)-decahydro-2,7-naphthyridin-2-yl]ethyl}pyrrolidin-2-one
(1S,5R)-6-[(3-fluoro-4-methoxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-methyl-2-[4-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperazin-1-yl]acetamide
7-(2,2-dimethylpropyl)-2-(1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
3-[2-(methoxymethyl)piperidine-1-carbonyl]benzene-1-sulfonamide
4-methyl-2-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)-1H-1,3-benzodiazole