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4-{4-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]phenyl}-2-methylbut-3-yn-2-ol
3-(4-fluorophenyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3-phenylpropanamide
[2,4,6-trimethyl-3-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)phenyl]methanol
N-(3-{[ethyl(oxan-4-ylmethyl)carbamoyl]amino}phenyl)cyclopentanecarboxamide
2-hydroxy-N-(1-hydroxybutan-2-yl)-N-(pyridin-3-ylmethyl)-6-(trifluoromethyl)pyridine-3-carboxamide
N-{[7-chloro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-4-acetamido-N-[2-(4-fluorophenyl)ethyl]benzamide
3-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-1-(2-oxo-2,3-dihydro-1H-indol-5-yl)urea
{6-[4-(2-chlorophenoxy)piperidine-1-carbonyl]pyridin-2-yl}methanol
5-[4-(benzyloxy)piperidine-1-carbonyl]-2-(propan-2-yl)-1,3-benzoxazole
(1R,5S)-N-(2-ethyl-3-methyl-1-benzofuran-7-yl)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(1R,5S,6S)-6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-3-azabicyclo[3.1.0]hexane
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(3-hydroxyphenyl)-N-methyl-5-oxopyrrolidine-3-carboxamide
4-{[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
N-methyl-3-[methyl({[4-(pyridin-2-yl)phenyl]methyl})amino]butanamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(2-hydroxypropyl)-9-[3-(methylsulfanyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
7-chloro-2-methyl-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-amino-4-(furan-3-yl)-6-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
(2S,4R)-4-amino-N-(propan-2-yl)-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}pyrrolidine-2-carboxamide
2-methyl-5-(2-oxo-2-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}ethyl)-3,4-dihydropyrimidin-4-one
N-cyclopentyl-1-{2-[2-(3-methoxyphenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
(3R,4R)-1-[1-(4-chlorophenyl)cyclopropanecarbonyl]-3,4-dimethylpyrrolidin-3-ol
methyl 3-[(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]propanoate
1-(2-methyloxolane-2-carbonyl)-4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine
1-(dimethylamino)-3-[2-({[2-(2-fluorophenyl)ethyl]amino}methyl)-4-methoxyphenoxy]propan-2-ol
2-(dimethylamino)-2-(4-methylphenyl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
N-(pentan-3-yl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-[2-(1,3-thiazol-4-yl)ethyl]-3-(1H-1,2,4-triazol-1-yl)adamantane-1-carboxamide
N-methyl-1-(2-phenylethyl)-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-amine
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]acetamide
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-methyl-N-[2-(4-methylphenoxy)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
1-(2,3-dihydro-1-benzofuran-7-carbonyl)-3-(4-methylphenoxymethyl)piperidine
2-cyclopentyl-N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-phenylacetamide
1-(2,6-dimethylpyridin-4-yl)-4-(1H-imidazol-4-ylmethyl)piperazine
(1R,6S)-9-methyl-3-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}-3,9-diazabicyclo[4.2.1]nonane
N-[4-({ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenyl]acetamide
4-[(diethylamino)methyl]-5-ethyl-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]furan-2-carboxamide
4-(1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
N2-(1-benzylpyrrolidin-3-yl)-N4-methylpyrimidine-2,4-diamine
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methyl-4-(pyridin-2-yl)pyrimidin-2-amine
1-[3-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
5-methyl-1-propyl-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1H-pyrazole-4-carboxamide
{4-[3-(3-fluorophenyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
5-benzyl-5-(piperidin-4-yl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}acetamide
2-[2-(benzyloxy)phenyl]pyridine-3-carbonitrile
N-[2-(dimethylamino)ethyl]-2,4-dimethyl-N-(oxolan-2-ylmethyl)pyrimidine-5-carboxamide
(3S,4S)-4-methyl-1-(2,3,4,9-tetrahydro-1H-carbazole-8-carbonyl)piperidine-3,4-diol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-4-chloro-N,1-dimethyl-1H-indole-2-carboxamide
3-[2-(4-chlorophenyl)morpholine-4-carbonyl]-1H-pyrazol-5-amine