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1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-1,4-diazepan-2-one
1-{2-[1-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1-ethyl-3-methyl-1H-pyrazole-5-sulfonamide
N-[(1-benzylpyrrolidin-3-yl)methyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
methyl 4-{4-[2-(1-benzyl-3-oxopiperazin-2-yl)acetyl]piperazin-1-yl}benzoate
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-{[3-(2-methylphenyl)phenyl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-4-(4-methoxyphenoxy)piperidine
(1-{[4-(furan-2-yl)phenyl]methyl}-4-[(4-methoxyphenyl)methyl]piperidin-4-yl)methanol
1-methyl-3-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-1,2,5,6,7,8-hexahydroquinolin-2-one
{2-ethoxy-5-[1-(oxolan-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]phenyl}methanol
(4aS,8aR)-6-[(2-fluorophenyl)methyl]-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
3-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(3-phenylpropyl)benzamide
1-{4-phenyl-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}ethan-1-one
({3-methoxy-2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)[(3-methyl-1H-pyrazol-5-yl)methyl]amine
N-[3-(1H-imidazol-1-yl)propyl]-2-methyl-N-(pyridin-4-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
(1R,5S)-6-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-6-azabicyclo[3.2.1]octane
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N,6-dimethylpyrimidin-2-amine
4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
4-fluoro-N-{2-[3-methyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]ethyl}benzamide
N3-[1-(furan-2-yl)ethyl]-4-oxo-1-(propan-2-yl)-N5-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
5-ethyl-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N,N-dimethyl-2-[methyl({4-[6-oxo-4-(pyridin-3-yl)-1,6-dihydropyrimidin-2-yl]phenyl}methyl)amino]acetamide
1-(4-{4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}phenyl)ethan-1-one
2-benzyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-benzoxazole-5-carboxamide
methyl 3-(2-methylbutanamido)-5-{[(3-methylphenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-(dimethylamino)-2-{2-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
1-(4-methylphenyl)-4-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]piperazin-2-one
methyl (2S,4R)-4-(2-cyclopropylquinoline-4-amido)-1-[(2,4-difluorophenyl)methyl]pyrrolidine-2-carboxylate
2-methyl-4-(4-methylphenyl)-1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperazine
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-[(E)-2-phenylethenesulfonyl]piperidin-4-ol
(1R,5R)-6-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
3-{[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]methyl}pyridin-2-amine
2-(2-{4-azaspiro[2.5]octan-4-ylmethyl}phenyl)-6-propyl-3,4-dihydropyrimidin-4-one
4-(6-methoxypyridin-3-yl)-6-methyl-2-propylpyrimidine
1-(6-ethyl-2-methylpyrimidin-4-yl)-N-[2-(1H-indol-3-yl)ethyl]piperidin-4-amine
6-methyl-3-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-1,4-dihydroquinolin-4-one
methyl 2-{[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]methyl}-1,3-oxazole-4-carboxylate
N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)pyrazolo[1,5-a]pyridine-2-carboxamide
N-methyl-1-phenyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-({2-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H-imidazol-1-yl}methyl)-1λ6-thiolane-1,1-dione
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]propanamide
(3aS,6aS)-N,N-dimethyl-5-[2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)acetyl]-octahydropyrrolo[3,4-b]pyrrole-1-carboxamide
N-{[1-(quinolin-4-ylmethyl)pyrrolidin-3-yl]methyl}cyclopropanesulfonamide
{1-[3-(furan-2-yl)propyl]piperidin-2-yl}methanol
N-cyclohexyl-3-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]propanamide
3-{[(5-methylthiophen-2-yl)methyl]amino}-N-[1-(pyridin-3-yl)propan-2-yl]benzamide
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(thian-4-yl)piperidin-3-yl]propanamide