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(1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)(pyridin-3-yl)methanol
N,N-diethyl-2-({1-[(4-methoxyphenyl)methyl]-2-oxo-4-[(1R,2R)-2-phenylcyclopropanecarbonyl]-1,4-diazepan-6-yl}oxy)acetamide
methyl 3-cyclohexyl-2-oxo-1-(1,3-thiazol-5-ylmethyl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
1-(4-ethylpiperazin-1-yl)-3-{1-[1-(6-methylpyridin-2-yl)propan-2-yl]piperidin-4-yl}propan-1-one
4-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperazin-2-one
N-(butan-2-yl)-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(thiophen-3-ylmethyl)propanamide
2-fluoro-N-(3-oxo-3-{2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}propyl)benzamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-3,6-dimethyl-1-benzofuran-2-carboxamide
N-{[8-(trimethylpyrimidin-4-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
4-[2-(4-hydroxyphenyl)acetyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
3-(cyclopentylsulfamoyl)-5-(1H-pyrazol-1-yl)benzoic acid
4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-chloro-N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)benzene-1-sulfonamide
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)-4-{[(2-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-8-(4-methyl-1H-pyrrole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(4aR,8aR)-4a-hydroxy-7-[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
1-benzyl-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidin-3-amine
2-(oxolan-2-yl)-1-(1-phenylmethanesulfonylpiperidin-4-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazole
2-{3-cyclopentyl-5-[(2,3-difluorophenyl)methyl]-1H-1,2,4-triazol-1-yl}acetic acid
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
3-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1-(2,4,6-trimethylphenyl)urea
1-{[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}piperidine-3-carbonitrile
1-[1-(oxan-4-yl)piperidine-4-carbonyl]-4-(1,3-thiazol-2-yl)piperazine
3-(4-hydroxyphenyl)-N-(2-methoxyethyl)-N-methylbenzamide
2-(azepan-1-yl)-1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}propan-1-one
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
1-[(3-hydroxyphenyl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
1-(methoxymethyl)-N-methyl-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]cyclobutane-1-carboxamide
3,6-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N2,N2,6-trimethyl-N4-[(5-methylpyrazin-2-yl)methyl]pyrimidine-2,4-diamine
N-{4-chloro-3-[3-(2-hydroxyethyl)-4-methylpiperazine-1-carbonyl]phenyl}acetamide
4-[(2-methyl-1H-imidazol-1-yl)methyl]-1-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(2-methoxyphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
5-chloro-2-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-3-phenyl-1H-indole
(1S,5R)-N-(3-ethylphenyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-(4-{[2-(hydroxymethyl)quinazolin-4-yl]amino}piperidin-1-yl)pyridine-3-carbonitrile
1-(cyclohexylmethyl)-3-cyclopropyl-5-(5-methyl-2H-1,2,3-triazol-4-yl)-1H-1,2,4-triazole
3-fluoro-N,5-dimethyl-N-[2-(phenylsulfanyl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
2-{[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidin-1-yl]methyl}-3,5-dimethoxybenzoic acid
7-chloro-4-[(3-ethyl-1H-pyrazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(3-fluorophenyl)-1-(4-methoxyphenyl)-4-(pyrrolidin-1-ylmethyl)-1H-pyrazole
1-(2-aminoethyl)-N-[3-(3,4-dimethylphenoxy)propyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
3-[2-(morpholin-4-yl)-2-oxoethyl]-4-[(3-phenoxyphenyl)methyl]piperazin-2-one
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-(4-methylpiperazin-1-yl)propan-1-one
3-[1-({2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)ethyl]adamantan-1-ol
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(thiophen-3-yl)propan-1-one
N-{[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl}-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-amine