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1-[6-hydroxy-4-(4-phenyl-1,3-thiazole-2-carbonyl)-1,4-diazepan-1-yl]ethan-1-one
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-2-phenylethane-1,2-dione
{4-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-1,4-oxazepan-6-yl}methanol
1-(diphenylmethyl)-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazine
1-(2-fluorophenyl)-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazine
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2,5-dimethylfuran-3-carboxamide
4-(1H-imidazol-1-ylmethyl)-1-{[2-(trifluoromethoxy)phenyl]methyl}piperidin-4-ol
9-[2-(methylsulfanyl)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]pyridine-2-carboxylic acid
3-[1-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-fluoro-3,4-dihydroquinazolin-4-one
1-(2-{[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}pyrimidin-4-yl)pyrrolidin-3-ol
5-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazol-2-yl}-2-phenyl-1,3-thiazole
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-4-ol
4-[5-methyl-4-(2-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaene
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-{[5-(methoxymethyl)furan-2-yl]methyl}piperazin-2-yl}ethan-1-ol
(3S,5R)-N3-(4-methylphenyl)-N5-[2-(3-methylphenyl)ethyl]piperidine-3,5-dicarboxamide
ethyl 1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-[(3-fluorophenyl)methyl]piperidine-4-carboxylate
2-[4-(isoquinolin-5-ylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-benzyl-N5-ethyl-N3-methyl-4-oxo-N3-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
1-(4-{3-[1-(2-fluoroethyl)-1H-pyrazol-3-yl]phenyl}phenyl)ethan-1-one
2-(4-methanesulfonylphenyl)-4-(piperidine-1-carbonyl)pyridine
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-(1-ethyl-5-oxopyrrolidin-3-yl)urea
6-ethyl-2-methyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]quinoline-4-carboxamide
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-sulfamoylthiophene-2-carboxamide
N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
(3R)-1-(4-ethyl-5-methylthiophene-3-carbonyl)-3,4,4-trimethylpyrrolidin-3-ol
N-cyclopropyl-2-oxo-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,2-dihydroquinoline-4-carboxamide
1-[4-(4-methoxyphenoxy)phenyl]-3-methyl-3-[3-(oxolan-2-yl)propyl]urea
2-methoxy-4-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carbonitrile
1-(2-phenylethyl)-N,5-bis(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1-[5-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-1,2,3,6-tetrahydropyridine
5-(4-methanesulfonylphenyl)-2-methyl-1,3-benzoxazole
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2-{5-[2-(morpholin-4-yl)pyrimidin-5-yl]-4-phenyl-1H-imidazol-1-yl}acetic acid
5,6-dimethyl-3-[1-(3-methylpyridin-2-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[2-(1H-imidazol-2-yl)ethyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-{3-[(1S,5R)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
{2-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]phenyl}methanol
7-methoxy-N,N-dimethyl-2-[2-(pyridin-3-yl)pyrimidin-5-yl]quinoline-4-carboxamide
N-methyl-5-(3-phenyl-1H-pyrazole-4-carbonyl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
3-(2-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-N-(2-methoxyethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{3-[2-(methylsulfanyl)ethyl]-5-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl}benzoic acid
2-methyl-4-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
3-(3-chloro-1,2-oxazol-5-yl)-1-[2-(morpholine-4-carbonyl)piperazin-1-yl]propan-1-one
N-(5-methyl-1,3,4-thiadiazol-2-yl)-4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
2-(2-phenyl-1H-imidazol-1-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
1-{1H-pyrrolo[2,3-b]pyridin-6-yl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-({1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
(3S,4R)-3-hydroxy-4-(hydroxymethyl)-N-(4-phenylphenyl)piperidine-1-carboxamide