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3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,4-dihydroquinazolin-4-one
8-methoxy-N-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
4-ethyl-1-methyl-3-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[4-(3,5-difluorophenyl)-1H-1,2,3-triazol-1-yl]-1-(1H-pyrazole-4-carbonyl)piperidine
2-(2-{[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]methyl}phenoxy)-1-(piperidin-1-yl)ethan-1-one
N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]thiophene-2-carboxamide
N-(1,4-dioxan-2-ylmethyl)-2-oxo-6-{[4-(pyrrolidin-1-yl)piperidin-1-yl]methyl}-1,2-dihydropyridine-3-carboxamide
5-{[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-(methylsulfanyl)pyrimidine
1-{3-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]propyl}-6-methyl-1,2-dihydropyridin-2-one
5-(4-methanesulfonylphenyl)-4,6-dimethyl-1H-pyrazolo[3,4-b]pyridin-3-amine
1-(5-chloro-2-methoxyphenyl)-3-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-3-(2-hydroxyethyl)urea
N-{[1-(3-fluoropropyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
1-(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-sulfonyl}benzoyl)pyrrolidine
2-{[4-(2-methoxyphenoxy)piperidin-1-yl]methyl}-6-methylpyridine
2-{4-[4-(4-ethoxy-3-methylphenyl)-4-oxobutanoyl]morpholin-3-yl}acetic acid
N-({1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}methyl)-2-(pyridin-4-yl)acetamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
2-methyl-6-[(4-phenylbutan-2-yl)amino]heptan-2-ol
1-(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-phenylpiperidine-4-carbonitrile
6-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoline
1-[2-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
4-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanoyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
methyl 4-{[({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}benzoate
N-(cyclohex-1-en-1-ylmethyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-tert-butyl-N-(furan-2-ylmethyl)-4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanamide
1-(3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propyl)-1H-1,2,3,4-tetrazole
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(1H-indazol-1-yl)ethan-1-one
9-[(2R)-2-hydroxy-2-(naphthalen-2-yl)acetyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
1-(2-{[2-(3-fluorophenyl)ethyl]amino}pyrimidin-4-yl)piperidin-3-ol
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-3-methoxypropan-1-one
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)[2-(2-methylphenoxy)ethyl]amine
(1S,5R)-3-(oxan-4-yl)-6-(3-phenyl-1,2-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-{[3,5-dichloro-4-(propan-2-yloxy)phenyl]methyl}-1λ6-thiomorpholine-1,1-dione
2-(2-acetyl-4,5-dimethoxyphenyl)-1-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]ethan-1-one
[(3R,4R)-1-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
2-(1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-2-yl)ethan-1-ol
4-[3-(4-ethylpiperazine-1-carbonyl)phenyl]-2-methylbutan-2-ol
N-[2-(3-methoxyphenyl)phenyl]-1-[(3-methylphenyl)methyl]piperidine-4-carboxamide
1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-4-[3-(pyrrolidin-1-yl)propyl]-1,4-diazepane
4-[4-ethyl-6-(thiophen-3-yl)pyrimidin-2-yl]morpholine
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-1,3-dimethyl-1H-pyrazole-4-carboxamide
N-cyclopentyl-4-oxo-4-[4-(oxolan-2-ylmethyl)piperazin-1-yl]butanamide
N-{2-[2-amino-7-methyl-4-(3-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-oxoethyl}acetamide
3-(3-hydroxy-3-methylbutyl)-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}benzamide
3-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-5-yl)-1-propyl-1-(pyridin-3-ylmethyl)urea
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,6-difluorobenzamide
2-amino-4-{methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]amino}quinazoline-6-carboxylic acid
(3R)-N-[3-(2-ethoxyethoxy)phenyl]-3-hydroxypyrrolidine-1-carboxamide
3-(2-fluorophenyl)-3-phenyl-N-[2-(1,3-thiazol-4-yl)ethyl]propanamide
4-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethylpiperazine-1-carboxamide