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N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)thian-4-amine
1-methyl-1-[(4-methyl-1H-imidazol-2-yl)methyl]-3-(1-methyl-1H-pyrazol-4-yl)urea
3-[2-(3-fluorophenyl)piperidine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-[5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
3-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
7-methyl-2-[(2-methyl-1-benzothiophen-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-{1-[1-(4-methylphenyl)propan-2-yl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
N-(3-methyl-1-oxo-1-{3-[(phenylsulfanyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}butan-2-yl)acetamide
1-{4-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]piperidin-1-yl}ethan-1-one
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
N-(furan-2-ylmethyl)-7-(1,3-thiazole-4-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3R,5S)-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
N-cyclopropyl-3-(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)propanamide
3-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-ylmethyl]benzonitrile
2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)-1-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one
2-(3-chloro-2,6-difluorophenyl)-1-[2-(ethylsulfanyl)ethyl]-1H-imidazole
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}pyridine-4-carboxamide
(3R,9aR)-8-(4-ethylbenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
5-(2,4-difluorophenoxymethyl)-N-[3-(morpholin-4-yl)propyl]-1,2-oxazole-3-carboxamide
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-{1-oxa-7-azaspiro[3.5]nonan-7-yl}pyridine-3-carboxamide
N-benzyl-6-ethyl-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(2S,4R,6S)-2-benzyl-6-{6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}oxan-4-yl]acetamide
2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}-N-{[3-(trifluoromethyl)phenyl]methyl}acetamide
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-2-propyl-1,3-thiazole-4-carboxamide
1-(2,2-diphenylethyl)-4-methyl-1,4-diazepan-5-one
3-(pyrazin-2-yl)-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}propan-1-one
1-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
3-{5-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
3-methoxy-2-[(3-propyl-1H-pyrazol-5-yl)formamido]propanoic acid
[(2,6-dimethoxyphenyl)methyl](methyl)[(3-methylpyridin-4-yl)methyl]amine
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[3-(methylsulfanyl)propyl]benzamide
N-(3-{3-[(3,4-difluorophenyl)amino]piperidine-1-carbonyl}phenyl)acetamide
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]thiophene-2-carboxamide
(1R,3S)-3-{[1-(2,5-difluorophenyl)cyclopropyl]carbamoyl}cyclopentane-1-carboxylic acid
5-(2,3-dihydro-1H-indene-1-carbonyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-(5-chloro-2-methoxybenzoyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
1-(1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}azetidin-3-yl)-2-methylpiperidine
N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3,4-trimethoxybenzamide
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propanamide
4-ethyl-6-{4-[3-(methoxymethyl)pyrrolidin-1-yl]piperidin-1-yl}-N,N-dimethylpyrimidin-2-amine
2,2-dimethylpropyl 5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carboxylate
3-fluoro-4-methoxy-N-[(5-methyl-1,2-oxazol-3-yl)methyl]benzamide
(1R,5R)-6-[2-(3-chlorophenyl)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
5-cyclopropyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-1,3-oxazole-4-carboxamide
N-cyclopropyl-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-amine
methyl (2R)-2-(4-hydroxyphenyl)-2-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}acetate
1-{1'-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
5-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]quinoline