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N-[1-(2-methoxyphenoxy)propan-2-yl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-tert-butyl-2-[3-(1H-imidazol-1-yl)propyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-methyl-3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
5-(2-fluorophenoxymethyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-1H-pyrazole-3-carboxamide
N-butyl-N-(furan-2-ylmethyl)-2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetamide
2-{[(3-phenylphenyl)methyl]amino}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-3-(piperidin-3-yl)benzamide
(1S,6R)-3-methyl-9-(2-methyl-5-propylpyrimidin-4-yl)-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[3-(4-fluorophenoxymethyl)-5-[(2-oxoazepan-1-yl)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
5-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-2,6-dimethyl-3,4-dihydropyrimidin-4-one
2-(4-methoxyphenyl)-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]acetamide
N-[2-(2-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
4-{2-[2-(2,3,4-trimethoxyphenyl)-1H-imidazol-1-yl]ethyl}-1,3-thiazole
2-methyl-5-phenyl-N-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(1,3-thiazol-2-ylmethyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N-methyl-2-(naphthalen-1-yl)benzamide
6-[3-(3-fluorophenoxymethyl)piperidine-1-carbonyl]-1-methyl-1H-indole
3-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]-3,9-diazaspiro[5.6]dodecan-10-one
N-cyclopentyl-4-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
methyl 5-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
2-(4,5-dimethyl-1H-imidazol-1-yl)-1-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
(3aS,6aS)-2-methyl-5-[2-(2,2,6,6-tetramethylpiperidin-4-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
methyl (2S)-2-({1-[3-(2-cyclopentylacetamido)phenyl]piperidin-4-yl}amino)-3-phenylpropanoate
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
5-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}methyl)-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
methyl({[(2R,5S)-5-[(1-methyl-1H-indazol-5-yl)methyl]oxolan-2-yl]methyl})(pyridin-3-ylmethyl)amine
(2-aminoethyl)bis(pyridin-4-ylmethyl)amine
N'-(2-ethoxyphenyl)-N-[(5-methylpyrazin-2-yl)methyl]propanediamide
methyl 3-({[1-(4-methoxyphenyl)cyclopentyl]formamido}methyl)-5-(pyrazine-2-amido)benzoate
{2-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-2-oxoethyl}urea
N-[(3S,4R)-1-[(2E)-3-phenylprop-2-en-1-yl]-4-propylpyrrolidin-3-yl]methanesulfonamide
2-[3-(2-chlorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]acetamide
2-(methylsulfanyl)-1-{4-[3-(morpholine-4-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyridin-3-ylmethyl)acetamide
N-[(2-chloro-6-fluorophenyl)methyl]-3-cyclohexyl-N-cyclopropyl-1H-pyrazole-4-carboxamide
N4-(oxolan-2-ylmethyl)-7-(1,3-thiazol-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-(furan-3-carbonyl)-4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidine
1-[2-(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-2-propylpyrrolidine-1-carboxamide
(1S,5R)-6-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-{[1-(methoxymethyl)cyclopentyl]methyl}-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
N5-ethyl-N3-methyl-4-oxo-1-(2-phenylethyl)-N3-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
(3S,5R)-1-[(4-methoxyphenyl)methyl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
5-(methoxymethyl)-N-[(4-methoxyphenyl)methyl]-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-4-({1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-1,3-oxazole
2-(1-methyl-1H-pyrazole-4-carbonyl)-N-[(5-methylfuran-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-1-methylazepane-2-carboxamide