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2-amino-6-(3-methyl-1-propyl-1H-pyrazol-4-yl)-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
2-amino-4-(3-chloro-4-methoxyphenyl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-(2,6-dimethylpyridin-4-yl)-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazine
N-ethyl-3-methyl-4-{[methyl(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)carbamoyl]amino}benzamide
N-[(3S,4R)-1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
3-{2-oxo-2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethyl}-1,3-oxazolidin-2-one
(3S,4S)-1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(dimethylamino)pyrrolidin-3-ol
2-amino-N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide
(2H-1,3-benzodioxol-4-ylmethyl)(prop-2-en-1-yl)(pyridin-2-ylmethyl)amine
3-methyl-3-phenyl-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-4-sulfamoylbenzamide
1-cyclohexanecarbonyl-N-(1H-indol-2-ylmethyl)pyrrolidine-2-carboxamide
1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N-methyl-N-{2-[2-(prop-2-en-1-yl)phenoxy]ethyl}-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1-cyclopentyl-5-oxopyrrolidine-3-carboxamide
ethyl({[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
2-(1H-1,3-benzodiazol-1-yl)-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]propanamide
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2,5-dimethylfuran-3-carboxamide
1-ethyl-8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(2-methyl-1,3-benzothiazol-5-yl)urea
N-[(3R,4S)-1-benzyl-4-cyclopropylpyrrolidin-3-yl]-4-cyanooxane-4-carboxamide
N-({1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
4-{4-[3-(3-methoxyphenyl)propanoyl]-2-oxopiperazin-1-yl}benzonitrile
4-[4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
1-benzyl-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-1H-pyrazole-4-carboxamide
2-(ethylsulfanyl)-5-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)pyrimidine
methyl 6-(but-2-ynoyl)-2-[(cyclopropylmethyl)(propyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-cyclohexyl-N-(quinolin-5-yl)piperazine-1-carboxamide
4-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(3-fluorophenyl)piperazin-2-one
5,7-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-4-(2-methylpyrrolidine-1-carbonyl)quinoline
7-fluoro-4-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydroquinolin-2-one
(2-methoxyethyl)({[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl})(propan-2-yl)amine
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methoxyethan-1-one
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N,5-dimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(5-ethyl-1,3-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]-1H-pyrazolo[3,4-d]pyrimidin-6-amine
1-(4-methoxyphenyl)-3-methyl-5-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine
2-[(3,4-difluorophenyl)methyl]-8-[2-(methylsulfanyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
3-methyl-6-[4-(pyrrolidine-1-carbonyl)phenyl]pyridazine
1-(4-methoxyphenyl)-3-methyl-4-(thiophene-3-sulfonyl)piperazin-2-one
(4aS,7aR)-1-(3-chloro-2-methylbenzoyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(morpholin-4-yl)propyl]-5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)piperidin-2-one
2-[(1S,5R)-3-(2-chloro-3-methylbenzoyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
2-(morpholin-4-yl)-1-[4-(2,4,6-trimethylphenyl)phenyl]ethan-1-ol
N-(2-hydroxyethyl)-3-(2-hydroxyphenyl)-N-{[4-(methylsulfanyl)phenyl]methyl}-1H-pyrazole-5-carboxamide
N,3-dimethyl-1-propyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
3-(6-methylpyridin-2-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(2-methylpyrimidin-5-yl)quinoline-4-carboxamide
N,1-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-(thiophen-2-yl)-1H-pyrazole-5-carboxamide