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N,2-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1-benzofuran-5-carboxamide
4-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-1-(2-methoxyethyl)pyrrolidin-2-one
1-benzyl-N3-butyl-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-ethyl-N-[1-(3-methylphenyl)piperidin-4-yl]pyrimidin-2-amine
3-benzyl-4-(2-methylfuran-3-carbonyl)piperazin-2-one
3-{[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]sulfamoyl}-N-phenylbenzamide
methyl 9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-3-[(2,3,6-trifluorophenyl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(3R,5S)-1-benzyl-N-butyl-5-[(4-methylpiperazin-1-yl)methyl]piperidine-3-carboxamide
{9-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(pyridine-2-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
5-(4-aminopyridine-2-carbonyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-methyl-5-{4-[2-methyl-2-(morpholin-4-ylmethyl)propyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
3-(1-methyl-1H-pyrazol-4-yl)-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
3-methyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]furan-2-carboxamide
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)-N-methylacetamide
3-(1-methylcyclopropyl)-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
4-ethyl-1-methyl-3-({1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[2-(4-fluorophenoxy)ethyl]-1-{[4-(methylsulfanyl)phenyl]methyl}-1,4-diazepan-5-one
1-[4-({[(3-fluoro-4-methylphenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(methanesulfonylmethyl)piperidine
(4aR,7aS)-1-butyl-4-(isoquinoline-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-({3-[1-methyl-3-(pyridin-3-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}methyl)morpholine
3-{2-oxo-2-[(2S)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-benzyl-3-(1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-methyl-2-(morpholin-4-yl)-N-[2-(oxan-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
4-(6-methoxypyridin-2-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[2-({[(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amino}methyl)quinolin-6-yl]acetamide
2-(benzyloxy)-1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]ethan-1-one
methyl 2-[(4-chlorophenyl)sulfamoyl]-6-(cyclohex-3-ene-1-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(4H-1,2,4-triazol-4-yl)benzamide
1-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-4-[(2-fluorophenyl)methyl]piperidine
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
ethyl 1-acetyl-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(1-methylpiperidin-3-yl)-1,3-oxazole-4-carboxamide
(8aS)-2-(pyridin-4-ylmethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
4-(1-{4-[6-(4-methylpiperazin-1-yl)pyridazin-3-yl]phenyl}ethyl)morpholine
N-[(1R,2R)-2-(dimethylamino)-2,3-dihydro-1H-inden-1-yl]-3-(3-hydroxy-3-methylbutyl)benzamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2-methyl-4-(2-methylphenyl)piperazine
1-[(3S)-3-(dimethylamino)azepan-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-[3-(dimethylcarbamoyl)-5-{[({4-[methyl(phenyl)amino]phenyl}methyl)amino]methyl}phenyl]pyridine-2-carboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{[(3R,4R)-4-(hydroxymethyl)-1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]pyrrolidin-3-yl]methyl}piperidin-4-ol
5-({5-[(N-methylmethanesulfonamido)methyl]furan-2-yl}methyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
4-[1-(4-propylpyrimidine-5-carbonyl)piperidin-4-yl]thiomorpholine
(1R,3s,6r,8S)-4-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}-4-azatricyclo[4.3.1.13,8]undecane
1-(diethylamino)-3-[2-methoxy-5-(1,4-oxazepan-4-ylmethyl)phenoxy]propan-2-ol
1-(2-ethylphenyl)-3-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]urea
(3aR,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-(2-propylpyridine-4-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(2H-1,3-benzodioxol-5-yl)-N-(furan-2-ylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxamide
1-(3-{5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)-3-(thiophen-2-yl)propan-1-one
N-[2-methyl-1-(pyrrolidin-1-yl)propan-2-yl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide