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5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-[2-(cyclohex-1-en-1-yl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
5-cyclohexaneamido-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
7-methoxy-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-{3-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(3-fluorophenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
1-[(4-fluorophenyl)methyl]-4-phenyl-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazole
(1R,5R)-6-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3aR,7aS)-2-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(1H-imidazol-1-yl)propan-1-one
1-[5-(1-methyl-1H-pyrazol-5-yl)furan-2-carbonyl]piperidine
1-(4-{[benzyl(ethyl)amino]methyl}-2-methoxyphenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
4,6-dimethyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
(2S)-2-[4-(2,3-dichlorophenyl)-1H-1,2,3-triazol-1-yl]-4-methylpentanamide
9-[(2-cyanophenyl)methyl]-N,N-diethyl-3,9-diazaspiro[5.5]undecane-3-carboxamide
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(3-methylpiperidin-1-yl)pyridine-3-carboxamide
3-(3-hydroxyquinoxalin-2-yl)-N-[2-methoxy-2-(thiophen-2-yl)ethyl]propanamide
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-[phenyl(pyridin-4-yl)methyl]-1,4-dihydropyridine-3-carboxamide
4-[(dimethylamino)methyl]-1-[4-(1H-pyrazol-3-yl)benzoyl]azepan-4-ol
methyl 3-(2,3-dihydro-1-benzofuran-5-ylmethyl)-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-3-(1H-pyrazol-1-yl)propanamide
1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]ethan-1-one
N-[(5-methylpyrazin-2-yl)methyl]-2-{4-[2-(pyridin-4-yl)acetyl]morpholin-3-yl}acetamide
2-ethyl-1-methyl-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
6-[3-(benzyloxy)propyl]-1,3-benzothiazol-2-amine
4-(2-amino-6-methylpyrimidin-4-yl)-1-ethyl-3-methylpiperazin-2-one
4-(2-methylpropyl)-3-{2-oxo-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethyl}piperazin-2-one
2-chloro-5-(1-{[3-(difluoromethoxy)phenyl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
3-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-1-(4-fluoro-3-methylphenyl)urea
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(morpholin-2-yl)ethan-1-one
5-(1,2-oxazolidine-2-carbonyl)-1-[2-(pyridin-2-yl)ethyl]piperidin-2-one
2-[3-(5-methylfuran-2-yl)-5-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepin-9-yl}-1H-1,2,4-triazol-1-yl]acetic acid
1-[(3S,5R)-3-(hydroxymethyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-methyl-1-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}piperidin-4-amine
(1S,4S)-2-(2-fluorophenyl)-5-[(3-methylthiophen-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
1-(2,2-dimethylpropyl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]pyrimidin-4-amine
N-[(3-methylphenyl)methyl]-2-[2-(propan-2-yloxy)propanamido]benzamide
3-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridin-3-yl}-N-methylformamido)-3-phenylpropanoic acid
2-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(2-fluorophenyl)ethyl)piperidin-1-yl]methyl}-5-methoxyphenol
3-{8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-(thiophen-2-ylmethyl)propanamide
2-methyl-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]thieno[3,2-d]pyrimidin-4-amine
5-{2-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]phenyl}-1H-1,2,3,4-tetrazole
4-{[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidin-1-yl]methyl}-N-(5-methyl-1,3,4-thiadiazol-2-yl)benzamide
2-fluoro-N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)benzamide
N-ethyl-5-{spiro[azepane-4,2'-chromene]-1-ylmethyl}pyrimidin-2-amine
1-[(5-fluoro-2-methoxyphenyl)methyl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
N-(1-{[(oxolan-2-ylmethyl)(propyl)carbamoyl]methyl}-1H-pyrazol-4-yl)-3-phenoxypropanamide
(1S,6R)-9-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide