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1-[3-(3-benzylpyrrolidine-1-carbonyl)phenyl]-1H-pyrazole
N-tert-butyl-2-(4-cyclopentylpyrimidin-2-yl)benzene-1-sulfonamide
N-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methyl)-4-methoxybenzene-1-sulfonamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-cyclopropyl-2-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-[3-(propan-2-yloxy)propyl]benzamide
3-(1-ethyl-1H-pyrazol-3-yl)-4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazole
3-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-1-[4-(methylsulfanyl)phenyl]urea
N-[2-hydroxy-2-(pyridin-4-yl)ethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-methoxypropan-1-one
3-methyl-7-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-(2-methoxyethyl)-1-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-3-(thiophen-3-ylmethyl)urea
2,6-dimethyl-N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]quinoline-4-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(3-methoxypropyl)piperazin-1-yl]ethan-1-one
3-{[(2-amino-5-ethylpyrimidin-4-yl)amino]methyl}-1,2,4-oxadiazole-5-carboxamide
N-(2-methoxyethyl)-N,6-dimethyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-cyclopentyl-4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-[4-(dimethylamino)phenyl]-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
1-[1-(4-methoxybenzoyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
N-{2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-oxoethyl}acetamide
4-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)piperazine-1-sulfonamide
(1S,5R)-6-[(2,4-difluorophenyl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N,3-dimethyl-N-pentyl-1-propyl-1H-pyrazole-4-carboxamide
[5-({3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)furan-2-yl]methanol
4-(2,3-difluoro-4-methoxybenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
(2S)-2-[2-(3,5-dimethoxyphenyl)-1H-imidazol-1-yl]propan-1-ol
4-({5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)imidazolidin-2-one
2-{1-[(3,4-difluorophenyl)methyl]-4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
N-(3-hydroxypropyl)-1-{1-[(3-phenoxyphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
(4aR,7aS)-1-acetyl-4-(1-benzofuran-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{1-[(2,2-difluoro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}piperidin-3-ol
N-[6-fluoro-2-oxo-4-(quinoxalin-2-yl)-1,2,3,4-tetrahydroquinolin-7-yl]-2-methylpropanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(quinolin-2-ylmethyl)piperidin-3-ol
2-[4-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperazin-1-yl]-1,3-benzothiazole
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]({[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl})methylamine
4-{[4-hydroxy-2-(4-methylphenyl)pyrimidin-5-yl]formamido}-N-methylbutanamide
5-(5-fluoro-2-methylphenyl)-2,4-dimethoxypyrimidine
1-{2-[(benzylamino)methyl]-5-methoxyphenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-heptylpiperazine
6-(1-cyclopropyl-5-oxopyrrolidine-3-carbonyl)-N,1-dimethyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
4-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonan-7-yl}-2,2-diphenylbutanenitrile
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-3-methylpyridine-2-carboxamide
N-[(3R,4S)-1-[(2-aminopyridin-3-yl)methyl]-4-propylpyrrolidin-3-yl]cyclobutanecarboxamide
2-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
ethyl 2,4-dimethyl-5-{methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]carbamoyl}-1H-pyrrole-3-carboxylate
3-(3-methoxybenzoyl)piperidine
1-[5-({5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1H-pyrazol-3-yl]ethan-1-one
6-[3-(morpholin-4-ylmethyl)phenyl]pyrazine-2-carboxylic acid
methyl 4-[(4-{2-[(2-methoxyethyl)carbamoyl]ethyl}piperidin-1-yl)methyl]benzoate
4-{3-[(3,4-dimethoxyphenyl)amino]piperidine-1-carbonyl}pyridin-2-amine