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[(3R,4R)-1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}isoquinoline
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-(5-propyl-1,3,4-thiadiazol-2-yl)piperidin-4-ol
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}pyridazine-3-carboxamide
1-phenyl-4-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butane-1,4-dione
N-(cyclohexylmethyl)-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
{1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
N4-{3-[cyclopentyl(methyl)amino]propyl}-5-methylpyrimidine-2,4-diamine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)pyrrolidin-3-yl]methanol
3-(oxolan-2-ylmethyl)-1-{4-[2-(pyridin-2-yl)ethoxy]phenyl}urea
3-(4-benzylpiperazine-1-carbonyl)-2-cyclopropyl-6-methyl-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
4-(2-chloro-6-methoxyphenyl)-6-methoxypyrimidin-2-amine
N-cyclopentyl-1-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
6-(benzyloxy)-1-cyclohexyl-4-(dimethyl-1,2-oxazole-4-carbonyl)-1,4-diazepan-2-one
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(2-phenoxyethyl)-1H-pyrazole-3-carboxamide
(2R,6R)-4-[2-methyl-2-(morpholin-4-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(1R,5R)-6-(cyclobutylmethyl)-3-(1,7-dimethyl-1H-indole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(5-{1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-imidazol-2-yl}furan-2-yl)methanol
1-methyl-3-(2-methylquinolin-8-yl)-1-(oxan-2-ylmethyl)urea
N-ethyl-3,4-dimethoxy-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
1-(furan-3-ylmethyl)-4-(2-phenoxyethyl)piperazine
N-(3-acetamido-4-fluorophenyl)-4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidine-1-carboxamide
(2R,6R)-4-({3-[(dimethylamino)methyl]phenyl}methyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-methyl-5-[(quinolin-8-yloxy)methyl]-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,2-oxazole-3-carboxamide
1-(2-{[(2-chloro-6-fluorophenyl)methyl](methyl)amino}ethyl)-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}urea
N-(2-{7-[(2-hydroxy-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
2-[(2-{[3,3-dimethyl-1-(pyridin-3-yl)butyl]carbamoyl}phenyl)amino]acetic acid
1-[3-(1H-imidazol-1-yl)propyl]-4-(1-methyl-3-phenyl-1H-pyrazol-4-yl)-1H-1,2,3-triazole
4-(furan-2-carbonyl)-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-ethyl-1-(2-phenylphenyl)urea
1-{4-[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-3-(thiophen-3-yl)propan-1-one
1-[(3-fluorophenyl)methyl]-5-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]piperidin-2-one
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2,2-dimethylpropyl)piperidine
6-methyl-4-(4-phenylazepane-1-carbonyl)-1,2-dihydropyridin-2-one
methyl 5-[2-(1H-1,2,4-triazol-5-yl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
3-(hydroxymethyl)-1-({2-[3-(piperidin-1-yl)propoxy]phenyl}methyl)pyrrolidin-3-ol
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(5-hydroxypyrazine-2-carbonyl)pyrrolidine-3-carboxylic acid
9-benzoyl-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[1-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)ethyl]-1,3,4-thiadiazol-2-amine
4-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-2,6-dimethylphenol
2-[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]-5-fluoro-1H-1,3-benzodiazole
3-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}(methyl)amino)-1-phenylpropan-1-ol
2-(1-ethyl-1H-pyrazol-4-yl)-N,7-dimethyl-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(4-fluoro-3-methoxyphenyl)methyl]pyrrolidin-3-yl]methanol
benzyl[(2-phenoxyethyl)sulfamoyl]amine
2-(2H-1,3-benzodioxol-5-yl)-1-(3-{[(dimethylsulfamoyl)amino]methyl}piperidin-1-yl)ethan-1-one