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2-(1H-indol-1-yl)-1-[2-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
2-methyl-4-[methyl(5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)amino]butan-2-ol
3-chloro-N-[2-(dimethylsulfamoyl)ethyl]-4-fluoro-1-benzothiophene-2-carboxamide
2-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-N-[1-(4-methylphenyl)ethyl]acetamide
[(3R,4R)-1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-[(2-ethoxypyridin-3-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
4-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepane-1-carbaldehyde
2-{5-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
2-[4-(hydroxymethyl)phenyl]-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
5-[(dimethylamino)methyl]-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-N-(propan-2-yl)furan-2-carboxamide
N-methyl-4-{[3-(thiophene-2-carbonyl)piperidin-1-yl]methyl}benzene-1-sulfonamide
N-[(3-chlorophenyl)methyl]-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
2-methyl-N-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)pyridine-3-carboxamide
1-(4-methoxyphenyl)-4-[5-(propan-2-yl)thiophene-3-carbonyl]piperazin-2-one
2-{2-[5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyrazine
N-[3-(3-fluorophenyl)phenyl]-1-(quinolin-5-ylmethyl)piperidine-4-carboxamide
N,N-bis(pyridin-3-ylmethyl)-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
2-(adamantan-1-yl)-1-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]ethan-1-one
1-ethyl-4-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}pyrrolidin-2-one
5-[({1-tert-butyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}methyl)sulfanyl]-1,3,4-thiadiazol-2-amine
1-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}imidazolidin-2-one
N-[(2-ethoxyphenyl)methyl]-N-ethyl-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
1-(1-benzylpiperidin-4-yl)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]piperidine-3-carboxamide
1-[5-(2,4-dimethoxyphenyl)-1,2,4-triazin-3-yl]-N,N-dimethylpyrrolidin-3-amine
2,2-dimethyl-5-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}thiomorpholin-3-one
4-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine
4-(hydroxymethyl)-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-ol
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[2-(methylsulfamoyl)ethyl]acetamide
1-{2-methyl-5-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]phenyl}imidazolidin-2-one
2-{[(1R,2R)-2-(benzyloxy)cyclopentyl]amino}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-cyclopropyl-3-{[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,2,4-oxadiazole
7-(cyclopropylmethyl)-2-[2-(3-fluorophenoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
(2R,6R)-1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
1-cyclopentyl-6-oxo-N-[3-(propan-2-yloxy)propyl]piperidine-3-carboxamide
1-[1-(4-fluorophenyl)ethyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
5-(3-acetylphenoxymethyl)-N-(2-hydroxyethyl)-N-methyl-1,2-oxazole-3-carboxamide
N-[(3R,4S)-1-acetyl-4-(propan-2-yl)pyrrolidin-3-yl]-2-chloro-3-methylbenzamide
N-[(2-tert-butyl-6-oxo-1,6-dihydropyrimidin-4-yl)methyl]acetamide
N-[(1-benzylpiperidin-3-yl)methyl]-1-cyclohexyl-1H-1,2,3-triazole-4-carboxamide
N-[3-(1H-indol-1-yl)propyl]piperidin-3-amine
1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-(2-ethoxyethyl)-5-[4-(hydroxymethyl)piperidine-1-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
N,N-dimethyl-5-(3-{1-[(3-methylpyridin-4-yl)methyl]-1H-pyrazol-3-yl}phenyl)thiophene-2-carboxamide
2-(1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidin-4-yl)-1,3-benzoxazole
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(3-propyl-1H-pyrazole-5-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[(1R,3R)-3-aminocyclopentyl]-2-[2-(benzyloxy)phenyl]acetamide
3-[1-(cyclohex-1-en-1-yl)ethyl]-1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]urea
1-({4-[2-hydroxy-3-(4-methylpiperazin-1-yl)propoxy]phenyl}methyl)-4-(hydroxymethyl)piperidin-4-ol
2-methyl-5-(3-{1-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-decahydro-1,6-naphthyridin-2-one