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N-(2-fluorophenyl)-3-{1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
{2-[7-(cyclobutylsulfamoyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-2-oxoethyl}urea
4-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-1-(2-methylphenyl)piperazin-2-one
methyl 3-{4-[2-(2,6-difluorophenyl)acetyl]-2-oxo-6-(pyridin-4-ylmethoxy)-1,4-diazepan-1-yl}propanoate
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-({1-[(1s,4s)-4-hydroxycyclohexanecarbonyl]pyrrolidin-3-yl}methyl)benzoic acid
1-[4-(pyridin-3-ylmethyl)piperazin-1-yl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
2-butyl-5-chloro-4-({3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1H-imidazole
2-({[5-(1-cyclopentanecarbonylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)ethan-1-ol
2-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]-N-ethylpyrimidin-4-amine
1-[1-(5-methyl-2-phenylfuran-3-carbonyl)piperidin-4-yl]piperidin-4-ol
4-benzyl-3-ethyl-1-(4-methyl-1H-pyrrole-2-carbonyl)-1,4-diazepan-5-one
2-[4-(3-hydroxyphenyl)piperidine-1-carbonyl]-5-methoxy-1,4-dihydropyridin-4-one
6-(4-chlorophenyl)-N-cyclopropyl-N-ethylimidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{2-[2-(3,4-dimethylphenyl)-1H-imidazol-1-yl]ethyl}-1,3-thiazole
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-2-(1H-pyrazol-1-yl)butanamide
1-[(1-benzylpyrrolidin-3-yl)methyl]-2-cyclopropyl-1H-imidazole
2-(2-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}ethyl)-1,2-dihydrophthalazin-1-one
1-[benzyl(methyl)amino]-3-{4-[(4-methoxypiperidin-1-yl)methyl]phenoxy}propan-2-ol
3-(3-fluorophenoxymethyl)-1-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(morpholine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[(4-phenoxyphenyl)methyl]-4-(pyrrolidin-3-yl)piperazine
4-[2-({4-benzyl-5-[1-(furan-2-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}sulfanyl)ethyl]morpholine
N-[(3R,4R)-3-hydroxy-1-(thiophen-3-ylmethyl)piperidin-4-yl]pyridine-3-carboxamide
8-(1,2-oxazole-3-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
5-{[1-(4-fluoro-3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-(methylsulfanyl)pyrimidine
5-methyl-N-[2-(piperidin-1-yl)ethyl]-6-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)thieno[2,3-d]pyrimidin-4-amine
1,5-dimethyl (2S)-2-{[1-(4,7-dimethylquinazolin-2-yl)piperidin-4-yl]formamido}pentanedioate
4-(3-methyl-1H-1,2,4-triazol-5-yl)-N-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)piperidine-1-carboxamide
2-{1-methyl-octahydropyrrolo[1,2-a]piperazin-2-yl}pyridine-3-carbonitrile
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)piperidin-2-one
6-cyclopentyl-2-(4-{[methyl(1H-pyrazol-5-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
[3-(hydroxymethyl)-4-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}phenyl]methanol
1-(2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidin-4-yl)pyrrolidin-3-ol
2-{4-[2-chloro-5-(trifluoromethoxy)phenyl]-1H-pyrazol-1-yl}-N-methylacetamide
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyridin-3-yl)ethane-1,2-dione
2-methyl-5-phenyl-N-[2-(1H-pyrazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]benzene-1,3-diol
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-3-methylpiperidine
3-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]-5-(dimethylsulfamoyl)-N-methyl-N-[1-(pyridin-4-yl)ethyl]benzamide
3-(1-acetylpiperidin-3-yl)-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-(1H-indol-3-yl)-N-{[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl}propanamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-(2-methyl-1H-imidazol-1-yl)acetamide
N-[3-(3-chlorophenyl)phenyl]-1-(1H-imidazol-2-ylmethyl)piperidine-4-carboxamide
3-(2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
N-(1,3-dihydroxypropan-2-yl)-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
2-amino-4-[(1,4-dioxan-2-ylmethyl)(methyl)amino]quinazoline-6-carboxylic acid
(4aS,7aR)-1-[(4-methylthiophen-2-yl)sulfonyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione