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5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-N,N-dimethyl-1,2,4-thiadiazol-3-amine
3-cyclohexyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-pyrazole-4-carboxamide
2-acetamido-N-{[4-(phenoxymethyl)thiophen-2-yl]methyl}acetamide
(3R,4R)-4-amino-1-[(5-methoxy-1H-indazol-3-yl)methyl]piperidin-3-ol
4-{2-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl}-N-methylbenzene-1-sulfonamide
5-{2-[(4aS,8aR)-1-(3-methylbutyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[1-(2,4-dimethoxyphenyl)ethyl]-N-methyl-2-(methylamino)pyridine-4-carboxamide
6-{2-[3-cyclopropyl-1-(3,5-dimethylphenyl)-1H-1,2,4-triazol-5-yl]ethyl}-2,3-dihydropyridazin-3-one
1-[(3S,4R)-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
3-{3-[3-(6-methoxypyrimidin-4-yl)phenyl]-1H-pyrazol-1-yl}propan-1-ol
3-chloro-4-fluoro-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1-benzothiophene-2-carboxamide
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]piperidine
methyl 5-[(3-methylbutyl)amino]-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-[(1-methylpiperidin-4-yl)methyl]pyrimidine
1-ethyl-N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]piperidin-3-amine
(1S,5R)-6-(2-methoxyethyl)-3-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[(2,3-dimethoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}-1,3-oxazolidin-2-one
7-fluoro-2-methyl-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}quinoline
N-{3-[2-(furan-3-yl)-1H-imidazol-1-yl]-2-methylphenyl}-3-methylbutanamide
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(2-hydroxy-2-phenylethyl)-N-methylpropanamide
N-methyl-1-(oxan-4-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
2-[5-(methoxymethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]-1H-1,3-benzodiazole
N-(6-methoxyquinolin-8-yl)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-(3-methylbutyl)-1,2-oxazole-3-carboxamide
1,3-dimethyl-N-(thiolan-3-yl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(3R,4R)-1-[(2-hydroxy-5-methoxyphenyl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
methyl[(4-{2-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl](thiophen-2-ylmethyl)amine
ethyl 1-(1H-1,3-benzodiazol-2-yl)-5-(morpholin-4-ylmethyl)-1H-pyrazole-4-carboxylate
3-methyl-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-2,3-dihydro-1,3-benzoxazol-2-one
3-{5-[(1S,3R)-3-aminocyclopentyl]-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-1-yl}benzoic acid
(2S)-2-{5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}propanamide
2-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}-5-fluoro-1H-1,3-benzodiazole
(4aS,8aR)-6-[benzyl(methyl)sulfamoyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(7-methyl-1-benzofuran-2-carbonyl)piperidine
N,N-diethyl-1-({1-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
N-(furan-2-ylmethyl)-N-methyl-3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
3,5-dimethyl-2-[4-(morpholine-4-carbonyl)piperazine-1-carbonyl]-1H-indole
(5R)-5-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
1-(5-methyl-1,3,4-oxadiazol-2-yl)-4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine
3-[(2-fluorophenyl)methyl]-5-(piperidin-4-yl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
3-ethoxy-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-2-(methylsulfanyl)pyridine-3-carboxamide
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3,5,7-trimethyl-1H-indole-2-carboxamide
2-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
3-(1-ethyl-1H-1,2,3,4-tetrazol-5-yl)-1-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]urea
4-cyclohexyl-1-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1H-1,2,3-triazole
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-(pyrrolidine-1-carbonyl)pyrazin-2-amine
1,3-dimethyl-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 1-{2-hydroxy-3-[4-({[(3-methyloxetan-3-yl)methyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate