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2-{4-[4-(4-fluorophenyl)-4-oxobutyl]-2-oxopiperazin-1-yl}benzonitrile
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-(oxolan-2-yl)thiophene-2-carboxamide
N-(2,4-dimethylphenyl)-4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidine-1-carboxamide
N-[(1R,2R)-2-acetamido-2,3-dihydro-1H-inden-1-yl]-5-propyl-1,2-oxazole-3-carboxamide
(1R,5R)-6-(cyclopropylmethyl)-3-(3-fluoropyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-1H-pyrazole-3-carboxamide
2-({[1-benzyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-5-methyl-1,3,4-oxadiazole
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-[(2,3,6-trifluorophenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]-3-(pyrazin-2-yl)propan-1-one
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
1-{2-[3-(butan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenyl}-1H-pyrazole
4-(dimethylamino)-N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]benzamide
2-{4-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperazin-1-yl}pyrazine
1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-4-(pyrimidin-2-yl)-1,4-diazepane
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylpropyl)acetamide
1-{7-[(3-methylphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}cyclopropane-1-carboxamide
N-[7-methoxy-2-oxo-4-(1,3-thiazol-2-yl)-1,2,3,4-tetrahydroquinolin-6-yl]butanamide
3-(1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}piperidin-2-yl)pyridine
6-(2-chlorophenyl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-2-methoxy-N-methylpyrimidine-5-carboxamide
2-(3-ethyl-2-imino-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
3-(3-hydroxyquinoxalin-2-yl)-1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]propan-1-one
7-[4-(benzyloxy)piperidine-1-carbonyl]-1,3-diazepane-2,4-dione
1-(2-chlorophenyl)-5-[1-(4-methyl-1H-pyrazol-1-yl)ethyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
4-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-fluoropyridine
(3aR,6aR)-2-(cyclobutylmethyl)-5-(2,3,4-trifluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1'-[2-hydroxy-2-(4-methoxyphenyl)acetyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,2-dihydroquinoxalin-2-one
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-3-(methanesulfonylmethyl)piperidine
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-[2-(pyridin-2-yl)ethyl]urea
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(pyridin-3-yl)propan-1-one
4-[(4-methyl-5-{1-[(4-methyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
9-methoxy-N-methyl-3-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-7-oxo-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-(2H-1,3-benzodioxol-4-ylmethyl)-3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-cyclopentyl-4-[4-(piperidin-3-ylmethyl)benzoyl]piperazin-2-one
N-(4-carbamoyl-3-chlorophenyl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane-9-carboxamide
2-methyl-1-{2-[3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]ethyl}-1H-imidazole
N-methyl-N-[(5-{3-methyl-6-oxo-4H,5H,6H,7H-[1,2]thiazolo[5,4-b]pyridin-4-yl}furan-2-yl)methyl]methanesulfonamide
N-[2-(4-phenylpyrimidin-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(3-chlorophenyl)-4-(quinoline-8-carbonyl)piperazin-2-one
N-methyl-2,4-dioxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-(2-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethyl)pyrrolidin-2-one
(1R,3S)-7-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
2-[4-(3-phenylprop-2-yn-1-yl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
6-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(3-chloro-4-methylphenyl)-3-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}urea
(3aR,6aS)-N-{1-[(2-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
1-(4-cyano-2-ethylphenyl)-3-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)urea