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2-(dimethylamino)-N-[(4,6-dimethylpyridin-3-yl)methyl]-2-(4-fluorophenyl)acetamide
5-[1-(3-methylpentanoyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
[(2-chloro-6-fluorophenyl)methyl]({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-[(2-chlorophenyl)methyl]-1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-fluoro-N-methylpyridine-4-carboxamide
1-[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-(cyclopropylmethyl)piperazine
4-{6-[4-(pyridin-3-ylmethyl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}morpholine
N-(1-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-(1H-imidazol-4-yl)-1H-imidazole
1-(4-methoxybenzoyl)-4-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperazine
methyl 1-benzyl-3-(furan-3-amido)-5-[(2-methylpropyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-3-methylthiophene-2-carboxamide
4-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]-2-methyl-5-propylpyrimidine
1-(2,6-dimethylpyridin-4-yl)-4-[3-(pyrrolidin-3-yl)benzoyl]piperazine
5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1-cyclohexyl-N-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
4-{[1-(furan-2-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
2-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-N,N-dimethylaniline
3-(morpholine-4-carbonyl)-N-[(1-phenylcyclohexyl)methyl]-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
1-[(2R)-oxolane-2-carbonyl]-3,3-diphenylpiperidine
2-(4-chlorophenyl)-2-[(1-cyclopropanecarbonylpiperidin-4-yl)formamido]acetic acid
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N,N-dimethylpiperidine-1-carboxamide
6-methyl-1-(oxolan-2-ylmethyl)-2-(2-phenylethyl)-3-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
N-[(2R,3R)-2-methoxy-1'-(3-phenylprop-2-ynoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
1-(4-{[8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}phenyl)ethan-1-one
2-{4-[(3-hydroxy-6-methylpyridin-2-yl)methyl]piperazin-1-yl}pyridine-3-carbonitrile
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-(methylsulfanyl)ethan-1-one
5,7-dimethyl-N-[3-(pyrrolidin-1-yl)propyl]pyrido[2,3-d]pyrimidin-4-amine
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
9-(1,2-oxazole-5-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N,6-dimethyl-2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-(dimethyl-1,2-oxazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(1-methylpiperidin-4-yl)-N-[3-(methylsulfanyl)propyl]piperidine-3-carboxamide
2-[2-(2,3-dihydro-1H-inden-1-yl)acetamido]-2-methylpropanoic acid
3-(2H-1,3-benzodioxol-5-yl)-N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
N-{1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]pyrrolidin-3-yl}acetamide
4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
2-(dimethylamino)-2-(3-methylphenyl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-methyl-1,4-diazepane
[(3R,5R)-1-(3-methyl-1-benzothiophene-2-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
N-methyl-6-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
N-[(3R,4S)-1-(carbamoylmethyl)-4-phenylpyrrolidin-3-yl]-4-cyanooxane-4-carboxamide
4-[2-(dimethylamino)-2-(4-methylphenyl)acetyl]-N,N-dimethylpiperazine-1-sulfonamide
(3S,5S)-1-(pyridin-4-ylmethyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-[(1-cyclooctylpyrrolidin-3-yl)methyl]acetamide
2-{[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]amino}pyridine-3-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
1-(carbamoylmethyl)-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]piperidine-4-carboxamide
4-{[(1S,5R)-6-[(dimethylcarbamoyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzoic acid