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8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(dimethyl-1,3-thiazol-5-yl)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
N-({5-[(5-acetylthiophen-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
2-(2H-1,3-benzodioxol-5-yl)benzamide
4-[(1-acetylpiperidin-4-yl)oxy]-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-methoxybenzamide
methyl 4-[2-(dimethylamino)-2-(4-methylphenyl)acetyl]piperazine-1-carboxylate
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-(pyrimidin-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N2-methyl-N2-[2-(2,3,6-trimethylphenoxy)ethyl]pyrrolidine-1,2-dicarboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-{4-[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
(1S,5R)-6-[2-(phenylsulfanyl)ethyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-ethyl-2-{1-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1H-imidazol-2-yl}pyridine
1-(4-{2-[(3-hydroxyphenyl)amino]-6-methylpyrimidin-4-yl}-1,4-diazepan-1-yl)-2-methoxyethan-1-one
5-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
1-(1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)pyrrolidin-2-one
N-(2-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}ethyl)acetamide
N-[(2R,3R)-2-methoxy-1'-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
4-{1-benzyl-5-[2-(oxolan-2-yl)ethyl]-1H-1,2,4-triazol-3-yl}benzamide
3-(3-methoxypropyl)-1-[1-(4-methylphenyl)cyclopropanecarbonyl]piperidine-3-carboxylic acid
ethyl 3-{[3-(azepane-1-carbonyl)-1-methyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propanoate
(4aR,8aS)-1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-6-(2-fluorobenzoyl)-decahydro-1,6-naphthyridine
2-benzyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1,3-thiazole-4-carboxamide
3-{2-[3-(2-ethylphenoxy)azetidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
(3R,4R)-1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3,4-dimethylpyrrolidin-3-ol
N,2,5-trimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1,3-oxazole-4-carboxamide
1-(2-cyclohexylethyl)-3-hydroxy-3-({[(2-methylpyridin-4-yl)methyl]amino}methyl)piperidin-2-one
N-[(1-cyclopentylpiperidin-3-yl)methyl]-5-methoxy-N-[2-(piperidin-1-yl)ethyl]furan-2-carboxamide
1-[(4-chlorophenyl)methyl]-N-methyl-N-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
1-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]-3-(pyridin-4-yl)propan-1-one
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl){[3-(trifluoromethyl)phenyl]methyl}amine
6-methyl-2-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carboxylic acid
5-(morpholin-4-ylmethyl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)furan-3-carboxamide
(1S,5R)-6-benzyl-3-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5-fluoro-3-methyl-2-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1H-indole
6,6-dimethyl-1-phenyl-N-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-methyl-2-(pyridin-4-yl)-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazole
(2S,4S)-N-ethyl-4-[2-(1H-imidazol-1-yl)acetamido]-1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidine-2-carboxamide
methyl (2S)-2-[(2-cyclohexyl-1,3-benzoxazol-6-yl)formamido]-2-phenylacetate
N-[2-(2,4,6-trimethylphenoxy)ethyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-4-yl)methanesulfonamide
4-chloro-1-methyl-N-[(1-methylpyrrolidin-3-yl)methyl]-1H-indole-2-carboxamide
4-(5-{[2-(furan-2-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)-1-methyl-1H-pyrazole
2-{[2-(1H-imidazol-1-yl)ethyl](methyl)amino}-2-[4-(propan-2-yloxy)phenyl]acetic acid
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-{thieno[3,2-d]pyrimidin-4-yl}piperazin-2-yl}ethan-1-ol
(3aS,6aS)-5-(4-aminopyrimidin-2-yl)-2-(cyclopropylmethyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl 6-{[methyl(1,2,3,4-tetrahydronaphthalen-1-yl)amino]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylate
4-(cyclopropylmethyl)-1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
N-{2-[({3-[2-hydroxy-3-(piperidin-1-yl)propoxy]-4-methoxyphenyl}methyl)amino]ethyl}acetamide