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[5-({3-[4-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}methyl)furan-2-yl]methanol
{[6-(4-fluoro-3-methylphenyl)pyridin-3-yl]methyl}dimethylamine
1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
(1R,5S,6S)-6-(azepane-1-carbonyl)-3-[2-methyl-2-(morpholin-4-yl)propyl]-3-azabicyclo[3.1.0]hexane
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-4,4,4-trifluoro-N-methylbutanamide
2-(4-methylphenoxy)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
6-ethyl-4-({methyl[2-(morpholin-4-yl)propyl]amino}methyl)-2H-chromen-2-one
2-(5-fluoro-2-methoxyphenyl)-2-[methyl(prop-2-en-1-yl)amino]acetic acid
4-chloro-3-fluoro-N-[(3-methyloxetan-3-yl)methyl]benzamide
4-{5-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
2-[1-benzyl-4-(3-chloropyridin-2-yl)piperazin-2-yl]ethan-1-ol
3-{5-[3-(1H-indol-3-yl)propyl]-3-methyl-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
N-[(3,4-dimethoxyphenyl)methyl]-N,1-dimethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{1-benzyl-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-5-yl}cyclopropane-1-carboxamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-N-[4-(furan-2-yl)phenyl]piperidine-3-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(propan-2-yl)acetamide
N-[(1R,2R)-2-(dimethylamino)-2,3-dihydro-1H-inden-1-yl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-[(4-methanesulfonylphenyl)methyl]-5-(4-methylpiperazin-1-yl)-2,3-dihydropyridazin-3-one
2-methyl-N-{3-[(pyridin-3-yl)amino]propyl}furan-3-carboxamide
(3S,4S)-4-cyclopropyl-1-[3-oxo-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]pyrrolidine-3-carboxylic acid
{1-[1-(morpholin-4-yl)cyclohexanecarbonyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
4-(1-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-3-yl)benzoic acid
N-(2-hydroxyethyl)-1-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(4S)-1-[2-(4-fluorophenyl)benzoyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(2-fluorophenoxymethyl)piperidine
1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}-4-phenyl-1,4-diazepane
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-3-(dimethylamino)benzamide
N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
{7-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-5-fluoro-2,3-dihydro-1-benzofuran-2-yl}methanamine
N-methyl-N-(quinoxalin-2-ylmethyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
3-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-1-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]urea
4-(4-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}piperazin-1-yl)quinazoline
4-(azocane-1-carbonyl)-2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-2,3-dihydro-1H-isoindol-1-one
3-ethoxy-1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]propan-1-one
3-{[1-benzyl-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-methyl-1H-indole
2-(2,3-dimethylphenoxy)-1-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
2-(2,3-dihydro-1H-inden-1-yl)-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]acetamide
7-(furan-2-ylmethyl)-N-[3-(1H-imidazol-1-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[3-(trifluoromethyl)benzoyl]piperidine
1-(3,4-difluorobenzoyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
3-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-1-(4-ethylpiperazin-1-yl)propan-1-one
(4aR,8aR)-7-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
1-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-indole-6-carboxamide
2-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
2-({[3-(prop-2-en-1-yl)-4-(prop-2-en-1-yloxy)phenyl]methyl}amino)acetamide
N-(2-methoxyethyl)-1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-enoyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
2-(4-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-N-methylpiperidine-3-carboxamide
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
2-(furan-2-yl)-N-[3-(3-methyl-1H-pyrazol-1-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine