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[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
4-[2-(4-fluorophenoxy)ethyl]-1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1,4-diazepan-5-one
methyl(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)(1,3-thiazol-2-ylmethyl)amine
3-[1-(1-cyclopropylethyl)-1H-pyrazol-5-yl]-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}urea
N-methyl-4-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}pyridin-2-amine
N-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]naphthalene-2-carboxamide
4-methyl-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)piperazine-1-sulfonamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-3-ol
N-{3-[(2-methoxyethyl)carbamoyl]-2-methylphenyl}-1-oxa-7-azaspiro[3.5]nonane-7-carboxamide
1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-[3-(trifluoromethyl)phenyl]piperazine
3-(1H-pyrazol-5-yl)-1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidine
2-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-(morpholin-4-yl)ethan-1-one
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-4-oxo-4H-chromene-2-carboxamide
N-methyl-4-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]pyridin-2-amine
4-ethyl-1-[2-(1H-imidazol-1-yl)ethyl]-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{[2-(1H-indol-3-yl)ethyl]amino}-N-(pyrazin-2-yl)acetamide
N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-2,3-dihydro-1H-indene-1-carboxamide
methyl(1,2-oxazol-3-ylmethyl){[2-(trifluoromethyl)phenyl]methyl}amine
(1S,6R)-3-(2,6-dimethylpyrimidine-4-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
(4S)-3,3,4-trimethyl-1-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-4-ol
4-(3,4-dichlorophenyl)-2-methyl-1H-imidazole
(2S)-N-[4-chloro-2-(trifluoromethyl)phenyl]-2-(methoxymethyl)pyrrolidine-1-carboxamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
4-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-(furan-2-ylmethyl)piperidine
1-(4-chlorophenyl)-N-{[1-(thian-4-yl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
1-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-3-(thiophen-2-ylmethyl)urea
3-hexyl-8-[2-(4-hydroxypiperidin-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S,4S)-N-ethyl-1-[(2-fluorophenyl)methyl]-4-(3,3,3-trifluoropropanamido)pyrrolidine-2-carboxamide
N-methyl-N-[3-(oxolan-2-yl)propyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[1'-(2-ethylpyridine-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
2-methyl-7-(6-methylpyridazin-3-yl)-N-(thiolan-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl](4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
3-(quinolin-6-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
2-(2-methoxyethyl)-8-{[4-(methylsulfanyl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-2-{5-methyl-3-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1H-pyrazol-1-yl}acetamide
1-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-3-(dimethyl-1,2-oxazol-4-yl)-1-methylurea
2-(4-fluorophenyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
4-(2-methoxyphenoxy)-1-[2-(1-methylpiperidin-2-yl)ethyl]piperidine
(5-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-2-ethoxyphenyl)methanol
4-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}-N-methyl-1,3-thiazol-2-amine
N-{2-[4-(dimethylamino)phenyl]ethyl}-2-(2-oxopiperidin-1-yl)acetamide
6-({[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}methyl)pyrimidin-4-ol
4-oxo-N-[(2-propyl-1,3-thiazol-4-yl)methyl]-4H-chromene-2-carboxamide
2-ethyl-4-phenyl-9-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecane
N-({1-[(2,3-difluorophenyl)methyl]pyrrolidin-3-yl}methyl)-2-(pyridin-2-yl)acetamide
3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-[3-(2-methoxyethoxy)phenyl]urea
3-methyl-N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]but-2-enamide