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(2S)-1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
methyl 9-(cyclopentyloxy)-3-(2,3-dimethoxybenzoyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(3-methyl-1H-pyrazol-1-yl)-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]propanamide
N,N-dimethyl-5-{[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methyl}pyridin-2-amine
1-{4-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-4-oxobutyl}piperidin-2-one
methyl 2-[(3,4-difluorophenyl)sulfamoyl]-6-(3,3-dimethylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
4-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-N-methylbenzene-1-sulfonamide
1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
4-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-3-fluoropyridine
N-[(2-chlorophenyl)methyl]-N-cyclopropyl-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)pyridine-3-carboxamide
2-{1-[2-(2-methylphenoxy)ethyl]-1H-imidazol-2-yl}benzoic acid
2-[(4-fluorophenyl)methyl]-4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}morpholine
N-(1-carbamoylcyclopentyl)-2,3-dihydro-1H-indene-1-carboxamide
1,6-dimethyl-N-[3-oxo-3-(pyrrolidin-1-yl)propyl]-1H-indole-2-carboxamide
2-methyl-3-[(pyridin-2-ylmethyl)amino]-N-(2,2,2-trifluoroethyl)benzamide
6,7-dimethoxy-3-({[(2-methoxyphenyl)methyl]amino}methyl)-N-methyl-N-(thiophen-3-ylmethyl)quinolin-2-amine
(2-ethoxy-5-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}phenyl)methanol
(benzylsulfamoyl)(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)amine
1-[2-(dimethylamino)ethyl]-4-ethyl-3-[1-(5-methylpyridine-3-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
[1-(1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanol
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1-methylazepane-2-carboxamide
1-[3-(methylsulfanyl)phenyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
4-(1,3-benzothiazol-2-yl)-N-[1-(propan-2-yl)-1H-pyrazol-5-yl]piperazine-1-carboxamide
4-methyl-3-(3-methylbutanamido)-N-(4H-1,2,4-triazol-4-yl)benzamide
2-(3-hydroxypiperidin-1-yl)-1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
1-[2-(3-methoxyphenyl)azetidin-1-yl]-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
N-[2-(4-fluorophenyl)ethyl]-N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-2,3,4-trimethoxybenzamide
2-(dimethylamino)-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-2-(2-methylphenyl)acetamide
1-(2-aminopyrimidin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-[5-(2-chlorophenyl)furan-2-carbonyl]-1,2-oxazolidin-4-ol
4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
8-(2-ethylpyrimidine-5-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
1-{3-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]phenyl}imidazolidin-2-one
N'-(4-methylphenyl)-N-[2-(1-methylpiperidin-3-yl)ethyl]propanediamide
2-[2-(4-methoxynaphthalen-1-yl)-1H-imidazol-1-yl]acetamide
2-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[1-(1-ethylpiperidin-4-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[2-(dimethylamino)pentyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(4-{4-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]piperazin-1-yl}phenyl)ethan-1-one
3-(1H-1,2,3-benzotriazol-1-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}propanamide
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-N-[2-(piperidin-1-yl)ethyl]pyridine-2-carboxamide
propan-2-yl 2-[(3,4-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxylate
N-(cyclohexylmethyl)-1-cyclopropyl-5-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
8-[2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)acetyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
2-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1H-indole
N-(9H-fluoren-9-yl)-6-({methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
5-cyclopropanecarbonyl-1'-(4-methylpyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]