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4-(3-hydroxy-3-methylbutyl)-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}benzamide
2-(2,4-difluorophenyl)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-3-(4-fluorophenyl)-1H-pyrazole-5-carboxamide
4-(4-fluorophenyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}oxane-4-carboxamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-phenyl-1H-pyrazole-5-carboxamide
2-methyl-4-(4-{[3-(pyridine-3-carbonyl)piperidin-1-yl]methyl}phenyl)butan-2-ol
4-[(3,4-difluorophenyl)methyl]-3-{2-[4-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
2-[(2,6-dichlorophenyl)methyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
8-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{4-[2-(methoxymethyl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}-N-methylethane-1-sulfonamide
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[4-(4-methyl-1H-pyrazol-3-yl)piperidin-1-yl]ethan-1-one
1-(4-chlorophenyl)-4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine
1-[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]-4-phenylbutan-1-one
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[2-(pyridin-3-yloxy)ethyl]amine
1-[5-({8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1-methyl-1H-pyrrol-3-yl]ethan-1-one
2-(2-methyl-1H-imidazol-1-yl)-1-[2-(2-phenylethyl)piperidin-1-yl]ethan-1-one
3-(1-methylpiperidin-3-yl)-1-[4-(9H-purin-6-yl)piperazin-1-yl]propan-1-one
2-{[4-(2,4,6-trimethoxyphenyl)-1H-1,2,3-triazol-1-yl]methyl}morpholine
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxane-4-carboxamide
4-methyl-3-(1H-pyrazol-4-yl)benzoic acid
3-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]-1,2-dihydroquinolin-2-one
3-{[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}benzonitrile
1-cyclopentyl-6-oxo-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
(4aS,7aR)-1-(1H-imidazol-2-ylmethyl)-4-(3-phenylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(4-fluorophenyl)methyl][(1-methyl-1H-1,3-benzodiazol-2-yl)methyl](pyridin-4-ylmethyl)amine
2-{4-[1-(4-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
7-(cyclopropylmethyl)-2-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]acetamide
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
(1S,5R)-6-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
5-acetamido-2-ethyl-1-(pyridin-3-ylmethyl)-N-[2-(1,3-thiazol-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
3-{[cyclohexyl(methyl)amino]methyl}-1-[(2-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
7-(cyclobutylmethyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(ethylsulfanyl)ethyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
(3R,4R)-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
4-fluoro-N-{2-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}benzamide
(4aS,8aR)-1-(3-methoxypropyl)-6-[(3-methyl-1,2-oxazol-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
1-{1-[(3-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}piperidin-4-ol
N-[2-(dimethylamino)ethyl]-5-[(3-hydroxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]phenol
N-[(2-ethoxypyridin-3-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-(carbamoylmethyl)-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
4-(1-{[3-(furan-2-yl)phenyl]methyl}piperidin-3-yl)pyrimidine
N,N-dimethyl-1-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-amine
methyl 3-benzamido-5-{[(3,4-difluorophenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}propanamide
4-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
3-chloro-N-[2-(phenylsulfanyl)ethyl]-N-(prop-2-en-1-yl)pyridine-4-carboxamide
3-[1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-4,5,6,7-tetrahydro-1,2-benzoxazole