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1-(2-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(6-methoxypyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(5-{1-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1H-imidazol-2-yl}thiophen-3-yl)prop-2-yn-1-ol
2-[4-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-methylpiperazin-2-yl]ethan-1-ol
4-{4-[(cyclopropylmethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}-6-methylpyrimidin-2-amine
1-{2-[(1-benzylpiperidin-4-yl)amino]pyrimidin-4-yl}piperidin-3-ol
N-cyclopropyl-2-(4-{[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}piperidin-1-yl)acetamide
4-(3-methyl-1H-pyrazole-5-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-methyl-4-(1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,2,5-oxadiazole
7-[(2,3-dimethoxyphenyl)methyl]-2-(2-methylpropyl)-2,7-diazaspiro[4.5]decan-6-one
methyl 3-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]propanoate
5-{[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-4-yl]methyl}-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
methyl (2S)-3-phenyl-2-({[(pyrazin-2-yl)carbamoyl]methyl}amino)propanoate
2-[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]-N-[1-(4-methylphenyl)ethyl]acetamide
(1S,5R)-6-(1-methyl-1H-pyrrole-2-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
{3-[(2-fluorophenyl)methyl]-1-(1-methyl-1H-indole-2-carbonyl)piperidin-3-yl}methanol
4-methyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-1H-imidazole-5-carboxamide
ethyl (4aS,8aR)-6-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylate
N-(2,3-dihydroxypropyl)-N-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
6-fluoro-2-{[(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amino]methyl}quinolin-4-ol
8-[2-(4-fluorophenyl)-2-(piperidin-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-3-(1H-pyrazol-4-yl)propan-1-one
1-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-(2-methoxyethyl)piperazine
4-(3-methoxyphenyl)-N-methyl-N-[2-(pyridin-4-yl)ethyl]benzamide
5-{[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]methyl}-N-propylpyrimidin-2-amine
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[2-(2-methylphenyl)pyrimidin-5-yl]methyl})amine
1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2,4-difluoro-3-methoxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
1-(2,5-dimethylphenyl)-3-phenyl-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1H-pyrazole
2,4-dimethyl-N-[4-(4-{[2-(pyridin-3-yloxy)ethyl]amino}piperidin-1-yl)phenyl]benzamide
8-fluoro-N-[2-(2-methylpropanesulfonyl)ethyl]quinoline-2-carboxamide
1-(2-methoxyphenyl)-4-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}piperazin-2-one
N-(2-methoxyethyl)-5-methyl-N-{[2-(2-methylphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}thiophene-2-carboxamide
1-methyl-4-{[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
3-[3-(4-fluorophenyl)oxolan-3-yl]-5-[(1H-1,2,4-triazol-3-ylsulfanyl)methyl]-1,2,4-oxadiazole
2-{5-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
ethyl 2-[9-(2,3-difluorobenzoyl)-3,9-diazaspiro[5.5]undecan-3-yl]acetate
(4aR,7aS)-1-(2-methylpropanoyl)-4-(pyrazine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(4-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
1-[(3,4-dimethylphenyl)methyl]-4-(3-fluorobenzoyl)piperazin-2-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,2-dimethyl-1,3-thiazole-4-carboxamide
N-(4-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-pyrrolo[2,3-b]pyridin-6-yl)piperidin-4-amine
4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-2-(thiophen-2-yl)-1,3-thiazole
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)(oxolan-3-ylmethyl)amine
1-{2-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[(4-methylphenyl)methyl]piperidin-3-ol
4-({4-[2-(pyridin-3-yl)piperidine-1-carbonyl]furan-2-yl}methyl)morpholine
3-methanesulfonamido-N-phenyl-5-[({[4-(propan-2-yl)phenyl]methyl}amino)methyl]benzamide
2-(3-methyl-1,2-oxazol-5-yl)-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)acetamide
2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-N-methylpyridine-3-carboxamide