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1-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-1-methylurea
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methylpiperidin-2-yl)methyl]amine
(2R)-1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-phenylpropan-1-one
N-methyl-3-(2-methylpropyl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1,2-oxazole-5-carboxamide
(5-{[1-(3-methoxypyrazin-2-yl)piperidin-4-yl]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
3,5-dimethyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
2-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]phenol
N-{2-[2-(pyridin-4-yl)-1H-imidazol-1-yl]ethyl}pyridine-3-carboxamide
3-(2-methoxyphenoxy)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}azetidine
1-({5-[2-(4-fluorophenoxy)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-methylpyrrolidine
2-(4-methylpentyl)-4-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]morpholine
2-methyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-1,3-benzoxazole-6-carboxamide
1-[(2-methylphenyl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
2-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]-4-methyl-1H-1,3-benzodiazole
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(4-methyl-1H-imidazole-5-carbonyl)pyrrolidin-3-yl]methanol
(3aR,7aS)-2-{2-[(4-methylpyrimidin-2-yl)oxy]hex-5-en-1-yl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
5-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-3-(thiophen-3-yl)-1H-pyrazole
2-[(cyclopropylmethyl)sulfanyl]-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
(3S,7S)-5-(2-acetylbenzoyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
methyl (2R)-2-[(5-methyl-4-{[(6-methylpyridin-2-yl)methyl]amino}thieno[2,3-d]pyrimidin-6-yl)formamido]propanoate
[3-(cyclopropylmethyl)-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]methanol
3-cyclopropyl-1-(1H-indazol-5-yl)-3-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
3-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-2-methylphenol
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-(thiophen-3-yl)propan-1-one
(oxolan-3-ylmethyl)(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-(1H-pyrazol-1-yl)benzamide
1-(2-{1-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
3-[4-(2-oxopyrrolidin-1-yl)phenyl]-1-[3-(phenylsulfanyl)propyl]urea
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,4-dimethyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carboxamide
5-methoxy-3-methyl-2-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-1H-indole
2-[2-(1-benzofuran-2-yl)phenoxy]propanamide
1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
3-{[1-(morpholin-2-ylmethyl)-1H-1,2,3-triazol-4-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
2-cyclopropanecarbonyl-8-[6-methyl-2-(methylamino)pyrimidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[3-(cyclohexyloxy)-2-hydroxypropyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-{5-[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}pyridazine
4-(2-methyl-1H-imidazol-1-yl)-1-{[(3-methylphenyl)methyl]carbamoyl}piperidine-4-carboxylic acid
2-(1H-pyrazol-1-ylmethyl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}-1,4-oxazepane
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,4-dimethyl-1H-imidazole-5-carboxamide
3-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
(2S)-N-(4-cyano-2-ethylphenyl)-2-(methoxymethyl)pyrrolidine-1-carboxamide
5-(cyclohexylamino)-1-ethyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-ethyl-3,5-dimethyl-4-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
3-(2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
N-(butan-2-yl)-1-(4-fluorophenyl)-N-(thiophen-3-ylmethyl)cyclopropane-1-carboxamide
methyl 4-{4-[2-(morpholin-4-yl)acetyl]piperazin-1-yl}benzoate
2-[2-({methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amino}methyl)phenoxy]acetic acid
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(1-methyl-1H-pyrrol-3-yl)acetamide
3-(hydroxymethyl)-1-{1-methyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-carbonyl}piperidin-3-ol