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N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-2-methyl-1-benzofuran-5-carboxamide
3-chloro-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}pyridin-2-amine
3-(1H-pyrazol-1-yl)-N-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
8-(2-aminopyrimidin-4-yl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
ethyl 4-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]piperidine-1-carboxylate
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-1-(propan-2-yl)piperidine-4-carboxamide
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-2,5-dimethyl-1,3-oxazole-4-carboxamide
N-[3-(4-methoxyphenyl)propyl]-6-[(1-methylpiperidin-4-yl)amino]pyridine-3-carboxamide
N-[3-(2-methoxybenzamido)phenyl]-3-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-methyl-4-[4-({methyl[1-(1,3-thiazol-5-yl)ethyl]amino}methyl)phenyl]butan-2-ol
1-(2-methylpropyl)-N-[(5-methylpyrazin-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
5-(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)-1-methyl-4-phenyl-1H-imidazole
7-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
N-(3-chloro-2-methylphenyl)-2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
2-[(2-hydroxyethyl)(methyl)amino]-2-[2-(methylsulfanyl)phenyl]acetic acid
2-(dimethylamino)-N-[2-(4-fluorophenyl)-1-{1-[3-(furan-2-yl)benzoyl]piperidin-4-yl}ethyl]-N-methylacetamide
1-({1-[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]piperidin-4-yl}methyl)pyrrolidin-2-one
4-ethyl-1-methyl-3-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(4-cyclobutanecarbonyl-1,4-diazepane-1-carbonyl)-5,6,7,8-tetrahydroquinoline
1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(oxan-3-yl)ethan-1-one
N-[2-(2,5-dimethylphenyl)ethyl]-3-[(2-fluorophenyl)formamido]propanamide
N-{3-[(2S)-2-amino-3-phenylpropanamido]phenyl}-4-methylbenzamide
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetamide
2-methyl-5-{2-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
4-[2-(methylsulfanyl)ethyl]-1-phenyl-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[3-(2-methoxyphenoxy)propyl]-N-methylmorpholine-2-carboxamide
1,3-dimethyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
1-{4-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}ethan-1-one
1-ethyl-6-{[3-(pyrimidin-4-yl)piperidin-1-yl]methyl}-1H-indole
6-[2-(2-aminoethyl)morpholin-4-yl]-2-(butylsulfanyl)pyrimidin-4-amine
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-(propan-2-yl)acetamide
3-(2-chlorophenyl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-5-methyl-1,2-oxazole-4-carboxamide
propyl (4aR,7aS)-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
1-[3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
1-{1-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]piperidin-4-yl}piperidine-4-carbonitrile
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
1-[(3-methoxyphenyl)methyl]-4-(7-methyl-1-benzofuran-2-carbonyl)piperazin-2-one
3-[(3S,4R)-1-benzyl-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(4-methoxyphenyl)propanamide
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)furan-2-carboxamide
1-(2-{1-[(5-fluoro-2-hydroxyphenyl)methyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
(5-{1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-phenyl-1H-imidazol-5-yl}furan-2-yl)methanol
2-hydroxy-2-methyl-1-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}propan-1-one
1-(furan-2-ylmethyl)-N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]piperidine-3-carboxamide
2,6-dimethyl-3-[3-(1H-pyrazol-1-yl)azetidine-1-carbonyl]quinoline
N-[(3S,4R)-4-(4-methylphenyl)-1-(quinoline-2-carbonyl)pyrrolidin-3-yl]acetamide
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[1-(3-methoxyphenyl)ethyl]methylamine
2-[5-(dimethyl-1,2-oxazol-4-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
(3S,9aR)-3-benzyl-8-[(2-fluorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide