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N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-[(piperidin-4-yl)amino]pyridine-3-carboxamide
3-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]-4-methylbenzoic acid
1-(2-cyclopentylacetyl)-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
{3-[2-(isoquinolin-5-yl)phenoxy]propyl}(methyl)amine
(1R,5S,6R)-3-(pyridin-2-ylmethyl)-N-[2-(thiophen-2-yl)ethyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
2-amino-6-(2,4-dichlorophenyl)-4-(oxolan-3-yl)pyridine-3-carbonitrile
6-{1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-3-yl}pyrimidin-4-ol
2-[(oxan-3-yl)amino]pyridine-3-carboxamide
(3aR,6aS)-5-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-3-[4-(furan-2-yl)butan-2-yl]urea
5-[3-(2-methylphenyl)piperidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidin-4-ol
5-{3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carbonyl}-4-propylpyrimidine
1-(methoxymethyl)-N-methyl-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}cyclopropan-1-amine
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-(pyrazin-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[2-(3-chlorophenyl)ethyl]-5-{2-[(2-methoxyethyl)amino]ethyl}pyrrolidin-2-one
1-{1-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}pyrrolidin-2-one
7-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(dimethyl-1,3-thiazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-aminoethyl)-N-[1-(furan-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
5-[2-(cyclohex-1-en-1-yl)acetyl]-1-(2-hydroxyethyl)-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(1-methoxybutan-2-yl)-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
3-cyclobutyl-4-[(1R)-1-(4-fluorophenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
6-methyl-5-[5-(oxan-2-yl)-1,2,4-oxadiazol-3-yl]-N-propyl-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
4-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-6-methylpyrimidin-2-amine
N-{[3-(furan-2-yl)phenyl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-methyl-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-[1-(pyrimidin-4-yl)ethyl]benzamide
(4aS,8aR)-1-(2-aminoethyl)-6-(thiophene-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-[4-(1H-1,3-benzodiazol-6-yl)phenyl]methanesulfonamide
4-{2-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
(4-{[1-(5-ethyl-1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]-4-phenyl-1H-imidazole-5-carboxamide
N-[3-(4-ethylpiperazine-1-carbonyl)phenyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(3,4-dimethoxyphenyl)-3-[2-(3-phenylpyrrolidin-1-yl)ethyl]urea
1-[4-(furan-3-ylmethyl)-6-hydroxy-1,4-diazepan-1-yl]-2-phenylethan-1-one
2,4-dimethyl-6-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
3,5-dimethyl-4-{5-[(3-methylthiophen-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-(prop-2-en-1-yl)-1H-pyrazole
9-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(cyclohexylamino)-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-one
N-(3-cyanophenyl)-2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-{[2-(dimethylamino)-4-methylpyrimidin-5-yl]formamido}-3-(furan-2-yl)propanoic acid
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(2-methoxyphenoxy)piperidine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(3S,4R)-4-methoxyoxolan-3-yl]benzamide
2-{[6-(2-methoxypyridin-3-yl)quinazolin-4-yl]amino}ethan-1-ol
(4aS,7aR)-1-(2-methoxy-3-methylbenzoyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(2-amino-6-methylpyrimidin-4-yl)-N-(2,3-dihydro-1H-inden-4-yl)piperazine-1-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]acetamide
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
(3S,4S)-1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
(1S,5R)-3-(4-chloro-2-fluorobenzoyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one