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N-(2,3-dihydro-1H-inden-1-yl)-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
3,4-dimethoxy-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
N3-(1-benzothiophen-2-ylmethyl)-N5-benzyl-N3-methyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-(4-chlorophenyl)-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
N-(pentan-3-yl)-1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
1-cyclopropyl-4-{4-[(pyridin-2-yl)amino]piperidine-1-carbonyl}pyrrolidin-2-one
5-(4-chlorophenoxy)-1,3-dimethyl-4-{1-propyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
2-(3-{1-[2-(piperidin-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyridine-3-carbonitrile
N-(5-chloro-2-methoxyphenyl)-3-{1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]piperidin-3-yl}propanamide
4-(1H-1,3-benzodiazol-1-yl)-1-[(3-methylphenyl)methyl]piperidine-4-carboxylic acid
2-amino-4-(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)-6-(1,3-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
(4aS,7aR)-1-[(4-chloro-2-fluorophenyl)methyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-[(2-fluorophenyl)methyl]-2-(1-methyl-1H-pyrazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(3S,4S)-1-{[4-ethoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
N-cyclooctyl-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
3-(2-fluorophenoxymethyl)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine
6-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2-propylpyrimidin-4-amine
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-3-(2-methylphenyl)-3-phenylpropanamide
3-ethyl-6-[3-(pyridin-2-yl)azetidine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]acetamide
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
N-methyl-2-(4-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)acetamide
({3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)diethylamine
(2R)-N-{2-[4-(dimethylamino)phenyl]ethyl}pyrrolidine-2-carboxamide
2-amino-7-{2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 6-(2-{[2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carboxylate
(1s,4s)-4-hydroxy-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}cyclohexane-1-carboxamide
1-{2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-oxoethyl}-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-methyl-2-oxo-8-(pyridine-3-sulfonyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-[2-(1-{[(2R)-1-ethylpyrrolidin-2-yl]methyl}-1H-1,2,3-triazol-4-yl)phenoxy]ethan-1-ol
(1R,7S)-3-[(4-fluorophenyl)methyl]-N-methyl-4-oxo-N-(1H-pyrazol-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-cyclopropyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-oxopyrrolidine-3-carboxamide
3-(adamantan-1-yl)-5-(oxolane-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-(oxolane-3-carbonyl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
1-{2-[3-(3-ethylphenoxy)azetidin-1-yl]-2-oxoethyl}-3-methyl-1,2-dihydroquinoxalin-2-one
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-butoxyethan-1-one
1-[(3S,4S)-3-hydroxy-4-(morpholin-4-yl)pyrrolidin-1-yl]-2-(1H-indol-3-yl)ethan-1-one
6-{4-[2-(pyridin-2-yl)ethyl]phenyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-[2-(methylsulfanyl)ethyl]-5-{[2-(trifluoromethyl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-(5,5-dimethyl-2,4-dioxoimidazolidin-1-yl)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methylacetamide
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-[(4,6-dimethylquinolin-2-yl)sulfanyl]propan-1-one
2,3,4-trifluoro-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}benzene-1-sulfonamide
(2S,4S)-N-methyl-4-[4-(2-{[(4-methylphenyl)carbamoyl]amino}propan-2-yl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)-6-[2-(pyrrolidin-1-yl)ethyl]pyridine-3-carboxamide
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}cyclohexanecarboxamide
3-methanesulfonamido-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
3-(1-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)-4-benzyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(4-{imidazo[1,2-b]pyridazin-6-yl}piperazin-1-yl)-2,5,6-trimethylpyrimidine