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2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)acetamide
8-chloro-2-{[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}quinoline
N-(3-methoxypropyl)-1,3-dimethyl-N-{[6-(thiophen-2-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-1H-pyrazole-5-carboxamide
1-(3-{4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine-1-carbonyl}phenyl)pyrrolidin-2-one
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
(3aR,6aR)-2-methanesulfonyl-5-[(3-methyl-1H-pyrazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{[methyl({[3-(2-{4-[4-(4-methylphenyl)benzoyl]piperazin-1-yl}ethoxy)phenyl]methyl})amino]methyl}pyrrolidin-2-one
3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-2-ethyl-6-methyl-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
(3R,5R)-5-(morpholine-4-carbonyl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]piperidine-3-carboxamide
6,7-dimethoxy-2-(pyrimidin-5-yl)quinazolin-4-amine
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-3-cyano-5-fluorobenzamide
1-(4,6-dimethylpyridine-3-carbonyl)-4-(2-methoxyphenyl)-2-methylpiperazine
(2R,3R)-3-amino-1'-(2-methoxypyridine-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}ethan-1-one
1'-[(3-chlorophenyl)methyl]-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
6-(4-fluorophenyl)-2-(4-hydroxypiperidine-1-carbonyl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
4-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]benzoic acid
1-(4-methoxyphenyl)-4-{3-[methyl(1-methylpyrrolidin-3-yl)amino]propanoyl}piperazin-2-one
1-[(4-methoxyphenyl)methyl]-4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-[1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]benzamide
1-{[(3S,4S)-1-(2-cyanobenzoyl)-3-hydroxypiperidin-4-yl]methyl}-3,3-diethylurea
5-chloro-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
(1S,2S)-2-[4-(3,5,7-trimethyl-1H-indole-2-carbonyl)piperazin-1-yl]cyclohexan-1-ol
4-[2-(2-fluorophenyl)ethyl]-3-(2-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 2-[benzyl(methyl)sulfamoyl]-6-[(2-hydroxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-benzyl-5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
4-{5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]pyrimidin-2-yl}morpholine
4-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
(4aS,7aR)-1-(3-cyclopropylpropanoyl)-4-(2-phenylethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 1-(2-methoxyethyl)-3-[2-(6-methylpyridin-2-yl)ethyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
2-({3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)pyridine
N-[(2-fluorophenyl)methyl]-3-{1-[3-(1H-indol-3-yl)propanoyl]piperidin-3-yl}propanamide
butyl({[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl})methylamine
(2S,3R)-2-{[2-(2-ethylphenoxy)ethyl]amino}-3-hydroxybutanamide
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-[2-(methylamino)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(methoxymethyl)-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
4-{[6-(3,4-dichlorophenyl)pyridin-3-yl]methyl}morpholine
1-(1,3-benzothiazol-2-yl)-N-(1H-imidazol-2-ylmethyl)piperidin-3-amine
(3S,4R)-4-(2-methylphenyl)-1-[2-(2-oxopiperidin-1-yl)acetyl]pyrrolidine-3-carboxylic acid
(3S,4R)-1-(1-benzoylpiperidin-4-yl)-4-phenylpyrrolidine-3-carboxylic acid
1-{[4-(benzyloxy)phenyl]methyl}-3-(pyrrolidin-1-yl)piperidine
8-[(3-hydroxyphenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazole
2-benzyl-N-[2-(2-oxopyrrolidin-1-yl)ethyl]-1,3-benzoxazole-5-carboxamide
2-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl)[(5-phenyl-1,2-oxazol-3-yl)methyl]amine
4-{4-[2-(methylsulfanyl)pyridine-3-carbonyl]piperazin-1-yl}quinazoline
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1-methyl-1H-pyrazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane