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methyl 2-[(4-chlorophenyl)sulfamoyl]-6-(4-methylpentanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
6-ethoxy-3-{[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]methyl}-1,2-dihydroquinolin-2-one
2-[3-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)phenoxy]acetamide
2-(2-fluoro-4-methoxyphenyl)-5-methyl-4-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1,3-oxazole
3,3-dimethyl-1-{[5-(quinolin-6-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-3-(1H-pyrazol-1-ylmethyl)benzamide
N-(1-benzylpyrrolidin-3-yl)-5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-{2-[(3,4-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}acetamide
2-[(4aR,7aS)-6,6-dioxo-4-[2-(propylsulfanyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
(3S,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidine-3-carboxylic acid
3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[4-(morpholin-4-yl)butyl]amine
2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-4-[(2-methyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
2-{[2-(1-ethyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}-1H-indole
1-{3-[(5-phenyl-1,2-oxazol-4-yl)formamido]propyl}piperidine-3-carboxamide
2-ethyl-4-phenyl-9-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-chloro-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}benzamide
N-[3-(4-methylpiperazin-1-yl)propyl]-4-(pyridin-3-yl)pyrimidin-2-amine
methyl 4-[5-(thiomorpholin-4-ylmethyl)-1,2,4-oxadiazol-3-yl]benzoate
1-ethyl-4-{[methyl({[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl})amino]methyl}pyrrolidin-2-one
3-[(3R,4S)-1-(2-ethylpyridine-4-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
3-(2-{[(5-methoxy-1H-indol-2-yl)methyl]amino}propyl)-3,4-dihydroquinazolin-4-one
ethyl 3,5-dimethyl-4-[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})carbamoyl]-1H-pyrrole-2-carboxylate
7-[(2,3-dimethoxyphenyl)methyl]-2-(pyridine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-(3-methoxyphenyl)-3-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]propanamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(4-methoxyphenyl)methyl]pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
(2S,4S)-4-amino-N,1-dimethyl-N-(2-methylprop-2-en-1-yl)pyrrolidine-2-carboxamide
1-{2-[5-(1-benzofuran-5-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrrolidin-2-one
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N,2,3,5-tetramethylpyrazolo[1,5-a]pyrimidin-7-amine
4-[5-({[2-(morpholin-4-yl)ethyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
[(4S)-4-amino-5-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-5-oxopentyl]urea
{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}(methyl)(quinoxalin-2-ylmethyl)amine
N-[3-(4-{[3-(pyridin-4-yl)propyl]amino}piperidin-1-yl)phenyl]-3-(trifluoromethyl)benzamide
1-(cyclopentylmethyl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
(2R,6S)-4-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-2,6-dimethylmorpholine
9-(oxolane-3-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[({[3-(2-{4-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperazin-1-yl}ethoxy)phenyl]methyl}(methyl)amino)methyl]pyrrolidin-2-one
N-(furan-2-ylmethyl)-N,1-dimethyl-5-{[(6-methylpyridin-2-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}morpholine-4-carboxamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]propanamide
N-(2H-1,3-benzodioxol-5-yl)-3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carboxamide
2-[8-chloro-2-(furan-2-yl)quinoline-4-carbonyl]-1,2-oxazolidin-4-ol
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-hydroxypropan-1-one
3-{3-[cyclohexyl(methyl)amino]propyl}-8-[(2S)-2-(methylamino)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]benzene-1-sulfonamide
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-6-methyl-1-(propan-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
8-{[2-(methylamino)pyridin-3-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-amino-1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}pyrrolidine-3-carboxylic acid