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N-butyl-2-(2-oxo-1,2-dihydropyridin-1-yl)-N-(pyridin-3-ylmethyl)acetamide
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)acetamide
2-cyclopropyl-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]pyrimidine-5-carboxamide
N-[(3,4-difluorophenyl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
5-chloro-N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]pyridine-2-carboxamide
2-methoxy-5-{[8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}benzoic acid
8-methyl-3-({methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
1-{4-[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-3-(2-methyl-1H-indol-1-yl)propan-1-one
2-{4-[(3,4-dimethylpiperazin-1-yl)methyl]phenyl}-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
4-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-2-ethyl-1-(propan-2-yl)piperazine
2-[4-(1-methylazepane-2-carbonyl)piperazin-1-yl]benzonitrile
5-[4-phenyl-5-(thiophen-3-yl)-1H-imidazol-1-yl]pentan-1-amine
6-methoxy-N4-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidine-2,4-diamine
5-chloro-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(2-cyclohexylethyl)-3-hydroxy-3-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)piperidin-2-one
2-[(3-hydroxy-2,2-dimethylpropyl)amino]-N-[1-(4-methylphenyl)ethyl]acetamide
3-({[(4-chlorophenyl)(phenyl)methyl]amino}methyl)-7-fluoro-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
N-{[3-(methylsulfanyl)phenyl]methyl}-N-(propan-2-yl)pyridine-3-carboxamide
(2S,4S)-4-amino-1-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
{4-[(3-fluorophenyl)methyl]-1-(6-methoxypyrimidin-4-yl)piperidin-4-yl}methanol
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-6-methoxyphenol
4-[1-phenyl-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]benzene-1-sulfonamide
7-(2,6-dimethoxybenzoyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(4aR,7aS)-1-benzyl-4-(pyridazine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
(3aR,6aR)-2-(prop-2-en-1-yl)-5-(quinazolin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrrolidine-3-carboxylic acid
2-(1-ethyl-1H-pyrazol-4-yl)-N,3,6-trimethyl-N-(propan-2-yl)quinoline-4-carboxamide
3-(2,2-dimethyloxan-4-yl)-3-ethyl-1-[3-(1H-pyrazol-5-yl)phenyl]urea
3-(4-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)propanamide
benzyl[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](oxolan-2-ylmethyl)amine
N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
1-(3-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-3-oxopropyl)piperidin-2-one
6-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1S,5R)-3-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(2-fluorophenyl)-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-sulfonamide
N-[4-(1H-indol-2-yl)phenyl]-1-[(2-methylpyrimidin-5-yl)methyl]piperidine-4-carboxamide
N-[(1r,4r)-4-hydroxycyclohexyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N,6-dimethyl-N-[4-(morpholin-4-yl)butyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
5-methyl-3-(3-{pyrazolo[1,5-a]pyridin-7-yl}phenyl)-1,2,4-oxadiazole
2-{[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}pyridine
1-(5-chloro-2-fluorobenzoyl)-2-(3-methoxyphenyl)piperidine
1-[4-(methylamino)pyrimidin-2-yl]-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
4-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
3-[(3R,4S)-1-(7-chloroquinolin-4-yl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
2-[2-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
[1-methyl-4-({2-[3-(piperidin-1-yl)propoxy]phenyl}methyl)piperazin-2-yl]methanol
2-[(pyridin-2-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(dimethylamino)-2-(4-methylphenyl)acetamide