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(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
(4S,4aS,8aR)-1-{imidazo[1,2-a]pyridine-6-carbonyl}-4-phenyl-decahydroquinolin-4-ol
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-4-hydroxy-2-(thiophen-2-yl)pyrimidine-5-carboxamide
1-(1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-1-oxopropan-2-yl)pyrrolidin-2-one
7-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-{2-[2-amino-3-cyano-6-(1H-pyrrol-2-yl)pyridin-4-yl]-4-chlorophenoxy}acetamide
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-benzyl-N-methyl-3-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-4-yl}propanamide
1-(5-ethyl-1,2-oxazole-4-carbonyl)-4-(2-methylphenyl)-1,4-diazepane
2-methyl-6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-4-(trifluoromethyl)pyridine
N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]pyridazine-3-carboxamide
(2S,4R)-4-amino-1-(2,1,3-benzothiadiazol-5-ylmethyl)-N-ethylpyrrolidine-2-carboxamide
2-ethyl-5-{[1-ethyl-3-(3-fluorophenoxymethyl)-1H-1,2,4-triazol-5-yl]methyl}-6-methyl-3,4-dihydropyrimidin-4-one
2-ethyl-6-methyl-5-(2-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}-2-oxoethyl)-3,4-dihydropyrimidin-4-one
1-(2-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
5-[1-(4-amino-5-methylpyrimidin-2-yl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
4-fluoro-N-({1-[2-(2-oxopiperidin-1-yl)acetyl]piperidin-3-yl}methyl)benzamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[(1-ethyl-1H-indazol-3-yl)methyl]acetamide
9-(1,5-dimethyl-1H-indole-2-carbonyl)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
1-(cyclopropanesulfonyl)-3,3-diphenylpiperidine
N-[2-(2-chlorophenyl)ethyl]-1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[1-(thiophen-3-yl)propan-2-yl]acetamide
N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-3-(1-methylpiperidin-3-yl)propanamide
4-({4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
1-[4-(methylsulfanyl)phenyl]-5-[1-(propan-2-yloxy)ethyl]-1H-1,2,4-triazole
2-(4-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}piperazin-1-yl)acetamide
3-{2-[5-(1-methyl-1H-indol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,3-oxazolidin-2-one
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)furan-2-carboxamide
3-(methoxymethyl)-1-{5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidine
N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-4-(3-hydroxy-3-methylbutyl)benzamide
dimethyl(3-{3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}propyl)amine
N-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
1-(1-cyclohexanecarbonylpiperidin-4-yl)-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2-(4-ethyl-2,3-dioxopiperazin-1-yl)-N-methylacetamide
4-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-methylimidazolidin-2-one
N-(butan-2-yl)-1-(methoxymethyl)-N-(thiophen-3-ylmethyl)cyclopropane-1-carboxamide
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]-2-(naphthalen-2-yl)ethan-1-one
N-(3-chlorophenyl)-9-oxa-2-azaspiro[5.5]undecane-2-carboxamide
N-benzyl-N-ethyl-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-amine
1-(3-fluorophenyl)-3-{1-[1-(3-phenylprop-2-ynoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
ethyl 2-chloro-5-{[2-(ethoxymethyl)pyrrolidine-1-carbonyl]amino}benzoate
1-[4-(6-aminopyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]-2-propoxyethan-1-one
3-fluoro-5-[4-oxo-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]benzonitrile
2-methyl-3-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,8-naphthyridine
1-(2-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)-1,2,3,4-tetrahydroquinolin-2-one
4-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-ylmethyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
4-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
N-[2-(2-ethoxyphenoxy)ethyl]-N,3,5-trimethyl-1H-pyrazole-4-carboxamide
N-(oxan-3-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
4-[(2-hydroxyphenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol