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4-[2-(4-chlorophenyl)morpholine-4-carbonyl]-2-methyl-1H-1,3-benzodiazole
N-cycloheptyl-3-{[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]amino}propanamide
4-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)piperazin-2-one
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(3-methoxypyrazin-2-yl)pyrrolidin-3-yl]methanol
3-benzyl-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(1-methylcyclopropanecarbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-{1-cyclopentyl-4-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
5-{[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]sulfonyl}-2-methoxy-N-methylbenzamide
(3R,4R)-3-cyclobutyl-1-[1-(2-methoxyethyl)piperidine-4-carbonyl]-4-methylpyrrolidin-3-ol
7-{2-[(1-methanesulfonylpiperidin-4-yl)amino]propoxy}-2H-chromen-2-one
4-ethyl-5-[2-(2-phenylethyl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
2-[(3-methoxyphenyl)sulfanyl]-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
N-{2-[7-(2H-1,3-benzodioxole-5-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclohexanecarboxamide
3-[4-(1-hydroxy-3-methylbutyl)piperidine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
2-(1-{[1-(5-chloro-2-methylbenzoyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
(2S,4R)-4-amino-N,N-diethyl-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)pyrrolidine-2-carboxamide
1-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(methylsulfanyl)propan-1-one
1-(2,3-dimethylphenyl)-N-(pyridin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)(2-phenylethyl)amine
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[2-(4-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]propanamide
5-{4-[(4-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
5-(1H-imidazol-1-ylmethyl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}furan-2-carboxamide
(2R,6S)-2,6-dimethyl-4-[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]cyclobutanamine
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-(3-fluorophenyl)piperazin-2-one
2-acetyl-8-[3-(pyridin-2-yl)propanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N,3,5-trimethyl-1H-indole-2-carboxamide
{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-cyclopropyl-2-hydroxy-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-[4-(trifluoromethyl)phenyl]acetamide
N,N-diethyl-2,7,8-trimethylquinoline-4-carboxamide
6-methyl-N-propyl-5-[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
2-{4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-6-(pyrrolidine-1-carbonyl)pyrazine
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
N-[(2-fluorophenyl)methyl]-2-[methyl(quinolin-5-ylmethyl)amino]acetamide
1-(6-aminopyrimidin-4-yl)-4-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1,4-diazepan-6-ol
(4aS,7aR)-1-[(2-chloro-6-fluorophenyl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-methyl-3-(2-oxo-2-{4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}ethyl)piperazin-2-one
ethyl 5-[3-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]-1H-imidazole-4-carboxylate
N'1-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]cyclopropane-1,1-dicarboxamide
[(4-cyclopropyl-5-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl)(1,2-oxazol-3-ylmethyl)amine
3,3-dimethyl-1-({5-[(1-methyl-1H-indol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
2-(dimethylamino)-2-(3-methylphenyl)-1-[(1s,5s)-7,10-dimethyl-3,7,10-triazatricyclo[3.3.3.01,5]undecan-3-yl]ethan-1-one
1-(4-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-4-[3-(pyridin-4-yl)propanoyl]-1,4-diazepan-2-one
3-cyclohexyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1H-pyrazole-4-carboxamide
2-(4-fluorophenoxymethyl)-4-hydroxy-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
2-{3-[(3S)-3-ethylmorpholine-4-carbonyl]phenyl}-4-methyl-1,2-dihydrophthalazin-1-one
3-methyl-3-[3-(1H-pyrazol-1-yl)propyl]-1-{3-[(trifluoromethyl)sulfanyl]phenyl}urea