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1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
{[(3S,4R)-1-(1-benzofuran-5-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
1-ethyl-4-{4-[4-(4-phenylpiperidin-1-yl)piperidin-1-yl]benzoyl}piperazine
N-(2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)pyridine-3-carboxamide
6-(cyclopropanesulfonyl)-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
1-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}butan-1-one
methyl (2S,4S)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-propanamidopyrrolidine-2-carboxylate
6-(4-ethylpiperazin-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
methyl N-{2-[4-(2-chlorophenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}carbamate
6-ethoxy-3-({methyl[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-[1-(4-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(2-hydroxyethyl)-N-methylacetamide
N3-(9H-fluoren-9-yl)piperidine-1,3-dicarboxamide
1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
3-(1-butyl-1H-imidazol-2-yl)-N-cyclopentylpiperidine-1-carboxamide
N-[1-(1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-3-methylbutanamide
2-{3-methyl-5-[2-methyl-5-(propan-2-yl)furan-3-yl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-(methoxymethyl)-1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
4-{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-5-phenyl-2-(pyridin-3-yl)pyrimidine
N-ethyl-5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(pentan-2-yl)furan-2-carboxamide
methyl 4-[5-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)-1,2,4-oxadiazol-3-yl]benzoate
(4aR,7aS)-1-acetyl-4-(3,4-dichlorobenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(2-amino-6-ethyl-5-methylpyrimidin-4-yl)(methyl)amino]-N-methylpropanamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-{[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]amino}-N-(propan-2-yl)pyridine-2-carboxamide
2,6-dimethyl-N-[2-(4-phenylpiperidin-1-yl)ethyl]imidazo[1,2-a]pyridine-3-carboxamide
[(4-ethylphenyl)methyl]({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-6-(propan-2-yl)pyrimidine
N-[(6-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyridin-3-yl)methyl]acetamide
2-[(3-fluorophenyl)methyl]-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}morpholine
N,5-dimethyl-N-(1,3-thiazol-4-ylmethyl)-4-[(thiophen-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-(3,5-dimethoxyphenyl)-2-[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]acetamide
2-(1H-indol-5-yl)-2-(morpholin-4-yl)acetic acid
2-(2,6-dimethoxyphenyl)-2-[4-(pyridin-4-ylmethyl)piperazin-1-yl]acetic acid
3-(4,4-difluoropiperidine-1-carbonyl)-N-(3-methoxypropyl)benzene-1-sulfonamide
6-methyl-5-[5-(oxan-4-ylmethyl)-1,2,4-oxadiazol-3-yl]-2-(pyrimidin-2-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
1-[(1R,5R)-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
4-{5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}morpholine
3-{[1-(3-chloro-4-hydroxybenzoyl)piperidin-4-yl]methyl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-hydroxy-1-(2-methoxyethyl)-3-{[methyl(propan-2-yl)amino]methyl}piperidin-2-one
N-cyclopropyl-4-({3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}sulfonyl)benzamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)oxan-4-amine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-8-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxamide
N3-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)piperidine-1,3-dicarboxamide
1-[(2-ethylpyrimidin-5-yl)methyl]-2-(3-fluorophenyl)azepane
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]propanamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
N-[2-(ethanesulfonyl)ethyl]-2,5-dimethyl-1,3-thiazole-4-carboxamide
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
5-[4-(aminomethyl)piperidin-1-yl]-2-[3-(1H-pyrazol-1-yl)propyl]-2,3-dihydropyridazin-3-one