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1-(cyclopropylmethyl)-4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperazine
(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
N-ethyl-2-[(isoquinolin-5-yloxy)methyl]-N-methyl-1,3-oxazole-4-carboxamide
2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine-3-carboxylic acid
3-(1H-indol-3-yl)-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}propanamide
(2R)-N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-hydroxy-2-phenylacetamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
3-tert-butyl-4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-({3-methyl-7-[2-(thiophen-3-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
2-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-1,3-thiazole
1-{4-[(4-fluoropiperidin-1-yl)methyl]-2-methoxyphenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
1-[(3R,4R)-4-(4H-1,2,4-triazol-4-yl)oxolan-3-yl]piperidine
2,3-dimethyl-7-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1H-indole
1-[(4-chlorophenyl)methyl]-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-6-oxopiperidine-3-carboxamide
2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
1-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazole
2-(3-chlorophenoxy)-1-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]ethan-1-one
4-(dimethylamino)-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]naphthalene-1-carboxamide
2,3,6-trimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]quinoline-4-carboxamide
methyl 1-(3,5-dimethyl-1-benzofuran-2-carbonyl)piperidine-4-carboxylate
4-[2-(1H-pyrazol-1-yl)ethyl]-1-[2-(pyrrolidin-3-yl)benzoyl]piperidine
1-{5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-pyrazol-3-yl}ethan-1-one
(3R,4R)-1-(2,3-dihydro-1H-indene-5-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-[3-(1,3-benzoxazol-2-yl)propyl]-2,1-benzoxazole-3-carboxamide
4-(2-methoxyethyl)-8-thia-4,6-diazatricyclo[7.6.0.02,7]pentadeca-1(9),2(7),5-trien-3-one
N-(2-methanesulfonamidoethyl)-2-methyl-1,3-benzoxazole-6-carboxamide
(3aR,6aR)-N-[2-(1H-imidazol-4-yl)ethyl]-2-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-(cyclopropylmethyl)-3-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
2-methoxy-1-[4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
(2S)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-[3-(pyridin-3-yl)propanoyl]pyrrolidine-2-carboxamide
3,5,7-trimethyl-2-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1H-indole
N-ethyl-1-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-N-(butan-2-yl)-N-cyclopentylacetamide
1-(2,3-dihydro-1H-inden-2-yl)-4-(1-methyl-1H-pyrrole-2-carbonyl)-1,4-diazepane
(2S,4R)-4-(dimethylamino)-1-(1H-imidazol-2-ylmethyl)pyrrolidine-2-carboxylic acid
(3aR,5R,6S,7aS)-2-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-octahydro-1H-isoindole-5,6-diol
4-{4-[2-(2-methoxyphenyl)acetyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
[(3R,4S)-1-[(2-chloro-4-fluorophenyl)methyl]-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
2-(2H-1,3-benzodioxol-5-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-1-yl]ethan-1-one
1-(1,1-dioxo-1λ6-thiolan-3-yl)-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-4-carboxamide
1-methyl-4-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-2-one
3-methyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-{3-[(trifluoromethyl)sulfanyl]phenyl}urea
(1S,5R)-6-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-(2-ethoxypyridin-3-yl)-2-methyl-6-propylpyrimidine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
1,4-dimethyl 2-{[1-(4-{[2-(morpholin-4-yl)ethyl]carbamoyl}phenyl)piperidin-4-yl]amino}butanedioate
1-(2,3-dihydro-1H-inden-5-yl)-2-(1-methyl-1H-imidazol-2-yl)-1H-imidazole
N-methyl-N-(2-methylpropyl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide