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4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
N-[2-(4-methoxyphenyl)ethyl]-N-[(4-methylphenyl)methyl]-2-(2-oxopiperidin-1-yl)acetamide
2,3-dimethyl-5-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carbonyl}benzene-1-sulfonamide
4-methyl-2-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-1H-1,3-benzodiazole
methyl[(4-phenyl-1,3-thiazol-2-yl)methyl]{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
N-[2-(3-{[(cyclopent-3-en-1-yl)carbamoyl]methyl}morpholin-4-yl)-2-oxoethyl]benzamide
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-3-(3-methylphenoxy)azetidine
5-(benzylamino)-N,N-dimethyl-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(1H-indole-6-carbonyl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
4-benzyl-3-ethyl-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-1,4-diazepan-5-one
3-(2-phenylethyl)-1-(9H-purin-6-yl)piperidine-3-carboxylic acid
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-[(1-methyl-1H-indol-4-yl)methyl]pyrrolidin-3-yl]methanol
2-(3-aminopropanoyl)-N-(1-phenylethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-(4-hydroxy-3-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}phenyl)acetamide
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyridin-3-yl)ethan-1-one
N-{2-[4-(4-methyl-1,4-diazepane-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}-2-(4-phenylphenyl)acetamide
1-(2-methoxyphenyl)-4-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}-1H-pyrazole
3-{2-[cyclohexyl(methyl)amino]ethyl}-8-(1-methylcyclopropanecarbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(2-methoxyphenyl)-3-(3,4,5-trimethoxyphenyl)-4H-1,2,4-triazole
2-(2-methoxyethyl)-9-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[1-(2,4-dimethylphenyl)-5-{4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl}-1H-1,2,4-triazol-3-yl]acetamide
2-(2-methoxyethyl)-8-(2-methyl-6-propylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
4,6-dimethyl-5-({3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrimidin-2-amine
N-(1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-2-carboxamide
4-(2H-1,3-benzodioxol-5-ylmethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-methyl-1H-1,3-benzodiazole
N-(4-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenyl)acetamide
[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
5-(2-benzyl-1,3-thiazol-4-yl)-3-methyl-1,2,4-oxadiazole
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-methyl-N-(quinolin-5-ylmethyl)propanamide
1-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methylbut-2-enamide
3-methyl-4-[2-oxo-2-(3-phenylpiperazin-1-yl)ethyl]-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-ethylmorpholine
6-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyridine-3-carbonitrile
({3-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)diethylamine
(2S,4R)-4-[(2,3-dihydro-1H-inden-2-yl)amino]-N-methyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
4-methoxy-2-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyrimidine
N-[2-(3-methoxyphenyl)ethyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
methyl 2-(1-{[4-(3-acetylphenyl)phenyl]carbamoyl}pyrrolidin-3-yl)acetate
2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-6-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,4-dihydropyridin-4-one
3,5-dichloro-4-methyl-N-[2-(pyrazin-2-yl)ethyl]benzamide
5-[1-(cyclopropylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-2-methyl-1,3-thiazole
N-[(6-hydroxypyrimidin-4-yl)methyl]-2-[(prop-2-en-1-yl)amino]benzamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
3-(2-fluorophenyl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
2-benzyl-5-(1,4-dioxan-2-ylmethanesulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine
6-methyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}imidazo[1,2-a]pyridine-2-carboxamide