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N-methyl-2-(3-methyl-1,2-oxazol-5-yl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-N-methylbenzene-1-sulfonamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(methylsulfanyl)propanamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-1,2,3-triazole-5-carboxamide
3-({2-[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazole-5-carboxamide
2-[(4-methoxyphenyl)methyl]-6-(morpholine-4-carbonyl)-1,3-benzoxazole
8-(2-methoxyacetyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-(4-methyl-5-phenylthiophene-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-methyl-5-phenyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1,2,4-oxadiazol-3-amine
3-{3-ethyl-5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazol-1-yl}-4-fluorobenzene-1-sulfonamide
1-(4-fluorophenyl)-4-[2-(pyridin-2-yl)pyrrolidin-1-yl]butane-1,4-dione
3-({4-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
3-(2-methyl-1H-imidazol-1-yl)-1-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one
1-cyclopropyl-4-({[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}methyl)pyrrolidin-2-one
6-(1-methyl-1H-imidazol-2-yl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]pyridazin-3-amine
N2-(4-methylphenyl)-6-(thiophen-3-yl)-1,3,5-triazine-2,4-diamine
1-[3-(4-phenoxybenzoyl)piperidin-1-yl]but-2-yn-1-one
(1r,4r)-4-({[3-(1H-pyrazol-1-ylmethyl)phenyl]formamido}methyl)cyclohexane-1-carboxylic acid
(1R,3S)-3-methoxy-7-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-7-azaspiro[3.5]nonan-1-ol
2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[2-phenyl-2-(piperidin-1-yl)ethyl]acetamide
6-ethyl-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-methylquinoline-4-carboxamide
4-{1-[1-(3-chloropyridin-2-yl)piperidin-4-yl]ethyl}morpholine
(3S,4S)-4-methyl-1-(5-phenyl-1,2-oxazole-4-carbonyl)piperidine-3,4-diol
2-[2-(1H-imidazol-4-yl)ethyl]-9-[2-(methylsulfanyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidin-1-yl)-2-oxoethyl]pyrrolidin-2-one
methyl 4-[4-(1-methyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]benzoate
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
N-(2-methoxyethyl)-4-methyl-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
4-(1-{1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
N-{2-[2-(methylcarbamoyl)ethyl]phenyl}-4-(pyridin-3-yloxy)piperidine-1-carboxamide
1-methyl-3-phenyl-N-[1-(pyrazin-2-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
N,N-dimethyl-4-[(6-methylquinolin-5-yl)methyl]piperazine-1-carboxamide
1-[1-(2,3-difluoro-4-methylbenzoyl)piperidin-4-yl]-3-phenylpropan-1-ol
(1S,5R)-3-benzyl-6-[2-(methylsulfanyl)pyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
4-cyclohexyl-3-[2-(2-hydroxyphenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S)-4-{3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxybenzoyl}-1,3-dimethylpiperazin-2-one
5-(4-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)-1,3,4-thiadiazol-2-amine
(2S,4S)-4-amino-1-[(2-hydroxy-6-methoxyquinolin-3-yl)methyl]-N-methylpyrrolidine-2-carboxamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxylic acid
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2,5-dimethyl-N-(oxolan-2-ylmethyl)benzamide
3-({[1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-3-yl]oxy}methyl)pyridine
2-{4-azaspiro[2.5]octane-4-sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-{5-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]thiophen-2-yl}ethan-1-one
9-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}-1,4,9-triazaspiro[5.5]undecan-5-one
4-({4-benzyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-5-chloro-1,3-dimethyl-1H-pyrazole
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[2-(diethylamino)ethyl]-N-methyl-1H-pyrazole-4-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-5-(oxolane-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
5-{1-[3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoyl]pyrrolidin-2-yl}-N-methylthiophene-2-carboxamide