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3,6-dimethyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
1-{4-[4-(3-chloro-4-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-methoxyethan-1-one
(1R,5S,6S)-6-({4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
N-[1-(hydroxymethyl)cyclopentyl]-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
4-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-1,3-oxazole-5-carboxamide
2-(7-fluoro-1H-indol-1-yl)-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
3-[(dimethylamino)methyl]-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidin-3-ol
1,3-dimethyl-6-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-(4-chloro-3-fluorophenyl)-N,N-dimethylpyridazin-3-amine
1-methyl-N-[(1-methylpiperidin-4-yl)methyl]-2,4-dioxo-N-(2-phenylethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-phenoxy-N-(1-{[(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]carbamoyl]methyl}-1H-pyrazol-4-yl)propanamide
4-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]pyridine
2-(dimethyl-1,2-oxazol-4-yl)-1-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}ethan-1-one
(2R,3R)-3-amino-1'-(2-propyl-1,3-thiazole-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-methyl-N-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-amine
(3S,4aS,8aS)-2-[(2S,4S)-4-amino-1-methylpyrrolidine-2-carbonyl]-N-tert-butyl-decahydroisoquinoline-3-carboxamide
2-benzoyl-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine
2-amino-N-[2-(4-ethylphenoxy)ethyl]-N,4-dimethyl-1,3-thiazole-5-carboxamide
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-(phenylamino)pyrimidine-5-carboxamide
1-[(5-chlorofuran-2-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane
5-(2-methoxyphenoxymethyl)-N-methyl-N-(thian-4-yl)-1H-pyrazole-3-carboxamide
4-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-2-(pyridin-3-yl)morpholine
[5-(1-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1H-imidazol-2-yl)furan-2-yl]methanol
(3R,4R)-1-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-4-(hydroxymethyl)piperidin-3-ol
N-(1-{1-[2-(2-chlorophenoxy)acetyl]piperidin-4-yl}-2-(2-methylphenyl)ethyl)-N-methylcyclobutanecarboxamide
N-{[4-(dimethylamino)oxan-4-yl]methyl}-2-ethylpyrimidine-5-carboxamide
2-methoxy-N-(1-propylpiperidin-4-yl)pyrimidine-5-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
1-(3-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}propyl)-1H-imidazole
2-[4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperazin-1-yl]-1,3-thiazole-4-carboxamide
N-{2-[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-(4-fluorophenyl)acetamide
1-[(4-oxo-1,4-dihydroquinolin-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-(7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)pyridin-1-ium-1-olate
4-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
2-[(3R,4R)-3-hydroxy-4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]quinoline-4-carboxylic acid
2-amino-6-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-4-(pyridin-3-yl)pyridine-3-carbonitrile
ethyl 4-[2-(methylamino)pyrimidine-5-amido]piperidine-1-carboxylate
2-[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenyl]pyridine
2-(4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)pyrimidine
5-ethyl-3-(1-hydroxy-4-methylpentan-2-yl)-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-(3-methoxypropyl)-9-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(4-chlorophenyl)methyl]-8-(1,2-oxazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-{[6-(pyrrolidin-1-yl)pyridazin-3-yl]oxy}ethan-1-one
3-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-3,9-diazaspiro[5.5]undecane
3-{8-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}propanoic acid
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,2,8-trimethylquinoline-4-carboxamide
2-{1-[(1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-2-amine