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(3S,4S)-1-[6-(2,5-dimethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-(propan-2-yloxy)pyrrolidin-3-ol
4-(1-ethyl-1H-imidazol-2-yl)-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]piperidine
N-(3-cyclohexyl-1H-1,2,4-triazol-5-yl)-2-(4-fluorophenyl)pyrrolidine-1-carboxamide
3-(azepane-1-sulfonyl)-5-[4-fluoro-3-(hydroxymethyl)phenyl]benzoic acid
(4aR,7aS)-1-ethyl-4-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
[7-(dimethyl-1,3-thiazol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-methyl-N-[3-(propan-2-yloxy)propyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(1-benzylpyrrolidin-3-yl)methyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
5-{[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-(3-{4-[2-(2-phenylethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine-1-carbonyl}phenyl)imidazolidin-2-one
1-{6-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]pyridin-3-yl}ethan-1-one
4-(5-propyl-1,3,4-oxadiazole-2-carbonyl)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
4-[(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-2-oxo-decahydro-1,6-naphthyridine-6-carbonyl]benzonitrile
2,6-dihydroxy-N-methyl-N-[2-(morpholin-4-yl)propyl]benzamide
7-[(3,4-dimethoxyphenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
4-(1H-imidazol-1-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
(3aS,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-[3-(pyridin-3-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 5-[2-(1H-indol-3-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-({2-[2-hydroxy-3-(pyrrolidin-1-yl)propoxy]-4-methoxyphenyl}methyl)piperidine-4-carbonitrile
5-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]isoquinoline
6-[2-(3-chlorophenoxy)propanoyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
3-{2-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
(2S)-3-phenyl-2-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}propanamide
(5S,9aS,9bS)-2-[(5-methylfuran-2-yl)methyl]-5-[1-(propan-2-yl)-1H-indol-3-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-methyl-N-(1,2-oxazol-3-ylmethyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
(2S)-1-{2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetyl}pyrrolidine-2-carboxamide
2-amino-6-{4-[(dimethylamino)methyl]thiophen-2-yl}-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)pyridine-3-carbonitrile
4-{4-[2-(dimethylamino)-2-(3-fluorophenyl)acetyl]piperazin-1-yl}benzonitrile
5-(propan-2-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrimidin-4-amine
(2S)-2-{2-[N-(4-methylphenyl)methanesulfonamido]acetamido}-3-phenylpropanamide
2-(benzyloxy)-N-[(3R,4S)-1-(carbamoylmethyl)-4-cyclopropylpyrrolidin-3-yl]acetamide
1-[({[7-fluoro-2-(3-methoxyphenyl)quinolin-3-yl]methyl}amino)methyl]cyclohexan-1-ol
4-cyclopentyl-N-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-3-oxopiperazine-1-carboxamide
5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]isoquinoline
ethyl 1-cyclobutyl-3-(2-phenoxyethyl)piperidine-3-carboxylate
(2S,4R)-4-[4-({[(5-fluoro-2-methylphenyl)carbamoyl](methyl)amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]propan-1-one
2,3-dimethyl-6-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-[2-(4-methoxyphenyl)ethyl]-2-methyl-N-[(1-methylpiperidin-4-yl)methyl]pyrimidine-5-carboxamide
(3R,4S)-3,4-dimethyl-1-[(5-propylfuran-2-yl)methyl]piperidin-4-ol
2-({2-[1-(oxane-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
4-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1λ6-thiomorpholine-1,1-dione
1-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-3-(1,3-dimethyl-1H-pyrazol-4-yl)urea
methyl 6-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}-3-[(2E)-3-phenylprop-2-enamido]thieno[2,3-b]pyridine-2-carboxylate
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
[3-propyl-1-(1,3-thiazol-4-ylmethyl)piperidin-3-yl]methanol
2-{[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]methyl}-3,4-dihydroquinazolin-4-one
5-(2H-1,3-benzodioxol-5-yl)-2-ethoxybenzamide