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N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-3,5-dimethyl-1-benzofuran-2-carboxamide
N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
2-[5-(dimethylamino)-1H-1,2,4-triazol-3-yl]-N,N-bis(propan-2-yl)benzamide
(3aS,6aS)-2-(cyclopropylmethyl)-5-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl (1R,3S,3aR,6aS)-3-(2-ethyl-4-methyl-1H-imidazol-5-yl)-5-methyl-1-(2-methylpropyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
4-(4-methyl-1H-pyrazol-1-yl)-1-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperidine-4-carboxylic acid
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-3-ol
N2-[(4,6-dimethylpyridin-3-yl)methyl]-N4-methylpyrimidine-2,4-diamine
1-(2-methoxyphenyl)-4-[2-(4-methylpiperidin-1-yl)propanoyl]piperazin-2-one
1-(2-methoxyethyl)-2-{[3-(1-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-imidazole
3-{[(adamantan-2-yl)amino]methyl}-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
1-(4,6-dimethylpyrimidin-2-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidin-4-amine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3-(piperidin-3-yl)benzamide
1'-[3-(1H-pyrazol-1-yl)benzoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(1H-1,3-benzodiazol-1-yl)-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(1-ethyl-1H-1,2,3-triazol-4-yl)urea
4-benzyl-3-ethyl-1-[2-(methylamino)acetyl]-1,4-diazepan-5-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-{[6-(morpholin-4-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-1,3-thiazole-5-carboxamide
1-(3-methoxybenzoyl)-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
1-ethyl-5-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[(4-chlorophenyl)methyl]-8-(6-hydroxyhexyl)-2,8-diazaspiro[4.5]decan-3-one
1-{2-[4-(2-amino-6-methylpyrimidin-4-yl)piperazin-1-yl]pyrimidin-4-yl}piperidin-3-ol
2-amino-4-[2-(ethylamino)pyrimidin-5-yl]-6-(1H-indol-3-yl)pyridine-3-carbonitrile
1-({5-[(2-ethoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]propanamide
4-benzyl-3-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(cyclopentylmethyl)-1-(2-methoxyethyl)-6-methyl-3-[4-(4-methylphenyl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-(1H-pyrazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N,N-bis(prop-2-en-1-yl)-2-[4-(pyridin-3-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]acetamide
1-[3-(4-phenylbenzoyl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-{[4-(5-ethylpyridin-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-4-methanesulfonylmorpholine
[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][4-(2-methyl-1H-imidazol-1-yl)butan-2-yl]amine
(1-{1-[4-(furan-2-yl)phenyl]piperidin-4-yl}pyrrolidin-3-yl)methanamine
2-(4-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}phenoxy)-1-(4-methylpiperidin-1-yl)ethan-1-one
5-ethyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-1,3,4-oxadiazol-2-amine
3-({4-[(carbamoylamino)methyl]-1H-1,2,3-triazol-1-yl}methyl)-N-cycloheptylpiperidine-1-carboxamide
N-cyclopentyl-4-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]-4-oxobutanamide
2-(4-{[3-(hydroxymethyl)-3-propylpiperidin-1-yl]methyl}phenyl)-6-(methoxymethyl)-3,4-dihydropyrimidin-4-one
9-(1H-imidazol-4-ylmethyl)-3,9-diazaspiro[5.6]dodecane
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(1-methyl-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]methanol
1-(3-chlorophenyl)-5-methyl-4-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanoyl]piperazin-2-one
5-(3-methylpiperidine-1-carbonyl)-N-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-cyclopentyl-4-{4-[(1,4-dioxan-2-ylmethyl)amino]piperidin-1-yl}benzamide
methyl 3-[(4-methoxy-3-methylphenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
8-methoxy-2-methyl-5-(1-methyl-1H-imidazol-5-yl)quinoline
4-(furan-2-yl)-2-[5-methyl-4-(3-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
N-cyclopropyl-N-(1H-indol-5-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[1-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2-phenylacetamide
2-({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane